Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50010519
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50095649((2E)-1-[(5-azido-6-chloropyridin-3-yl)methyl]-N-ni...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataKi:  50nMAssay Description:Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed