Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50035160
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataKi:  8nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366737(CHEMBL1793971)
Affinity DataKi:  10nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366726(CHEMBL1793982)
Affinity DataKi:  20nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366733(CHEMBL1793973)
Affinity DataKi:  30nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366749(CHEMBL1793983)
Affinity DataKi:  50nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366736(CHEMBL1793972)
Affinity DataKi:  70nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366727(CHEMBL1793981)
Affinity DataKi:  100nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366729(CHEMBL1793969)
Affinity DataKi:  200nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366752(CHEMBL1793970)
Affinity DataKi:  250nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366728(CHEMBL1793978)
Affinity DataKi:  400nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366750(CHEMBL1793987)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50218940(CHEMBL1793991)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366738(CHEMBL1793985)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366738(CHEMBL1793985)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366726(CHEMBL1793982)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366745(CHEMBL1793989)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50218931(CHEMBL1793992)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366745(CHEMBL1793989)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366749(CHEMBL1793983)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366741(CHEMBL1793974)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366733(CHEMBL1793973)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50218958(CHEMBL1793984)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366731(CHEMBL1793990)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366739(CHEMBL1793994)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50218957(CHEMBL1793967)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366736(CHEMBL1793972)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366726(CHEMBL1793982)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366731(CHEMBL1793990)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366729(CHEMBL1793969)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366734(CHEMBL1793967 | CHEMBL1793980)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366746(CHEMBL1793976)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366732(CHEMBL1793979)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366743(CHEMBL1793968)
Affinity DataIC50:  33nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366741(CHEMBL1793974)
Affinity DataIC50:  34nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366727(CHEMBL1793981)
Affinity DataIC50:  45nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366728(CHEMBL1793978)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366749(CHEMBL1793983)
Affinity DataIC50:  67nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366733(CHEMBL1793973)
Affinity DataIC50:  86nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366743(CHEMBL1793968)
Affinity DataIC50:  91nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366735(CHEMBL1793993)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366751(CHEMBL1793977)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366744(CHEMBL1793988)
Affinity DataIC50:  175nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366747(CHEMBL1793975)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366729(CHEMBL1793969)
Affinity DataIC50:  257nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366736(CHEMBL1793972)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366728(CHEMBL1793978)
Affinity DataIC50:  419nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM198122(HC toxin)
Affinity DataIC50:  430nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366727(CHEMBL1793981)
Affinity DataIC50:  444nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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