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Found 7 Enz. Inhib. hit(s) with all data for entry = 50010622
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096859(CHEMBL135551 | Octadecanoic acid {2-[3-(2,3-dimeth...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096860((E)-3-Biphenyl-4-yl-N-{2-[3-(2,3-dimethyl-phenylsu...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096861(CHEMBL440905 | Heptadecanoic acid {[3-(2,3-dimethy...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096862((9Z,12Z)-Octadeca-9,12-dienoic acid {2-[3-(2,3-dim...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096860((E)-3-Biphenyl-4-yl-N-{2-[3-(2,3-dimethyl-phenylsu...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant prenyl protein-specific protease Rce1 expressed in Sf9 cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096861(CHEMBL440905 | Heptadecanoic acid {[3-(2,3-dimethy...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant prenyl protein-specific protease Rce1 expressed in Sf9 cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCAAX prenyl protease 2(Homo sapiens (Human))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096862((9Z,12Z)-Octadeca-9,12-dienoic acid {2-[3-(2,3-dim...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of recombinant prenyl protein-specific protease Rcel expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed