Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50010636
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096921(3-[4-(1-Methyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096922(3-(1-Methyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096914(8-Methyl-3-(1-methyl-1H-indol-5-yl)-8-aza-bicyclo[...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096915(3-(1-Ethyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]octa...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096913(3-(1-Ethyl-1H-indol-5-yl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096916(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096926(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicycl...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096919(8-Methyl-3-[4-(1-methyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096918(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096923(3-[4-(1,5-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096920(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096925(3-[4-(1-Methyl-5-phenyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096924(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-a...)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096917(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-methy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096914(8-Methyl-3-(1-methyl-1H-indol-5-yl)-8-aza-bicyclo[...)
Affinity DataIC50:  0.75nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096913(3-(1-Ethyl-1H-indol-5-yl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096915(3-(1-Ethyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]octa...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096922(3-(1-Methyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]oct...)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096916(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataIC50:  32nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096920(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-...)
Affinity DataIC50:  58nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096921(3-[4-(1-Methyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataIC50:  614nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096919(8-Methyl-3-[4-(1-methyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataIC50:  703nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096923(3-[4-(1,5-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataIC50:  825nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096926(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicycl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096925(3-[4-(1-Methyl-5-phenyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096917(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-methy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096924(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-a...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50096918(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataIC50:  1.47E+3nMAssay Description:Displacement of [125I]-RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed