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Found 32 Enz. Inhib. hit(s) with all data for entry = 50048512
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  2nMAssay Description:Binding affinity to rolipram binding site in isolated rat brain by rolipram binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219180(CHEMBL347429)
Affinity DataIC50:  70nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataIC50:  110nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219184(CHEMBL157897)
Affinity DataIC50:  110nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataIC50:  180nMAssay Description:Binding affinity to rolipram binding site in isolated rat brain by rolipram binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219177(CHEMBL347478)
Affinity DataIC50:  240nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219181(CHEMBL346928)
Affinity DataIC50:  430nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219177(CHEMBL347478)
Affinity DataIC50:  491nMAssay Description:Binding affinity to rolipram binding site in isolated rat brain by rolipram binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219180(CHEMBL347429)
Affinity DataIC50:  755nMAssay Description:Binding affinity to rolipram binding site in isolated rat brain by rolipram binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219185(CHEMBL157550)
Affinity DataIC50:  950nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219185(CHEMBL157550)
Affinity DataIC50:  950nMAssay Description:Binding affinity to rolipram binding site in isolated rat brain by rolipram binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219181(CHEMBL346928)
Affinity DataIC50:  1.01E+3nMAssay Description:Binding affinity to rolipram binding site in isolated rat brain by rolipram binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  1.80E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219193(CHEMBL158266)
Affinity DataIC50:  2.31E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219178(CHEMBL157832)
Affinity DataIC50:  3.05E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219199(CHEMBL352034)
Affinity DataIC50:  3.34E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219189(CHEMBL436416)
Affinity DataIC50:  4.48E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219198(CHEMBL156232)
Affinity DataIC50:  4.75E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219183(CHEMBL157204)
Affinity DataIC50:  5.15E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219191(CHEMBL156928)
Affinity DataIC50:  5.75E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219194(CHEMBL158202)
Affinity DataIC50:  6.11E+3nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219195(CHEMBL423595)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219179(CHEMBL156010)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219196(CHEMBL157308)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219197(CHEMBL440917)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219182(CHEMBL156054)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219192(CHEMBL156742)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219187(CHEMBL156985)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219186(CHEMBL155536)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of phosphodiesterase 4 from rat liver at 0.3 uM (not determined)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219190(CHEMBL154936)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219188(CHEMBL346569)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration for inhibitory activity against phosphodiesterase 4 from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50219184(CHEMBL157897)
Affinity DataIC50:  2.34E+4nMAssay Description:Binding affinity to rolipram binding site in isolated rat brain by rolipram binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed