Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50010831
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataKi:  0.0700nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataKi:  0.0800nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataKi:  0.230nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataKi:  0.260nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(CHEMBL411117 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  0.270nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(CHEMBL410166 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  0.460nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataKi:  0.520nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataKi:  2.21nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(CHEMBL413455 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  2.30nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(CHEMBL413426 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  4.80nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(CHEMBL386823 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  5nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(CHEMBL386823 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  5.80nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(CHEMBL386823 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  11.3nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(CHEMBL438914 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  25.7nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(CHEMBL411117 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  33.4nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(CHEMBL265391 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  34.8nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataKi:  55nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(CHEMBL413455 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  65nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(CHEMBL410166 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  65.5nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(CHEMBL413426 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  99nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataKi:  115nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(CHEMBL413426 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  464nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(CHEMBL410166 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  624nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(CHEMBL411117 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  662nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(CHEMBL413455 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  822nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50034121(CHEMBL386823 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099197(CHEMBL411117 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  1.04E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099199(CHEMBL413426 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  1.12E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(CHEMBL438914 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  1.42E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(CHEMBL265391 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  1.65E+3nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099201(CHEMBL413455 | Ile-Asn-Pro-Cys-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  2.34E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(CHEMBL438914 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  2.40E+3nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(CHEMBL265391 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  3.74E+3nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099202(CHEMBL265391 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  5.08E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099203(CHEMBL438914 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataKi:  7.10E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099200(CHEMBL410166 | Ile-Glu-Pro-Dpr-Tyr-Arg-Leu-Arg-(CH...)
Affinity DataKi:  7.89E+3nMAssay Description:Affinity for cloned Y5 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataEC50:  0.160nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y4 receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataEC50:  2.5nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y4 receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataEC50:  983nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y2 receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataEC50:  0.460nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y2 receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50099198(CHEMBL429531 | Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-Gly...)
Affinity DataEC50:  7.89nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y5 receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers

Curated by ChEMBL
LigandPNGBDBM50409214(CHEMBL2110365 | GR-231118)
Affinity DataEC50:  2.05E+3nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y5 receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed