Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50011092
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102217(3-[5-(4-Fluoro-phenylcarbamoyl)-1-oxy-pyridine-2-s...)
Affinity DataIC50:  32nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102229(6-Benzenesulfonyl-N-(4-fluoro-phenyl)-1-oxy-nicoti...)
Affinity DataIC50:  90nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102225(CHEMBL39740 | N'-(3-[2,2']Bithiophenyl-5-yl-6,7-di...)
Affinity DataIC50:  110nMAssay Description:Compound binding was evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human C-X-C chem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102216(6-Ethanesulfonyl-N-(4-fluoro-phenyl)-1-oxy-nicotin...)
Affinity DataIC50:  130nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102219(CHEMBL61835 | N-(4-Fluoro-phenyl)-6-methanesulfony...)
Affinity DataIC50:  130nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102226(CHEMBL58619 | N-(4-Fluoro-phenyl)-1-oxy-6-phenylme...)
Affinity DataIC50:  280nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102218(CHEMBL61655 | N-(4-Fluoro-phenyl)-1-oxy-6-(propane...)
Affinity DataIC50:  400nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102230(6-Cyclopentanesulfonyl-N-(4-fluoro-phenyl)-1-oxy-n...)
Affinity DataIC50:  460nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102221(6-Chloro-N-(4-fluoro-phenyl)-1-oxy-nicotinamide | ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102224(6-Chloro-N-(4-iodo-phenyl)-1-oxy-nicotinamide | CH...)
Affinity DataIC50: >2.00E+4nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102228(CHEMBL60578 | N-Benzhydryl-6-chloro-1-oxy-nicotina...)
Affinity DataIC50: >2.00E+4nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102227(6-Chloro-N-cyclohexyl-1-oxy-nicotinamide | CHEMBL6...)
Affinity DataIC50: >2.00E+4nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102220(CHEMBL293139 | N-(4-tert-Butyl-phenyl)-6-chloro-1-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102223(6-Chloro-N-(4-methoxy-phenyl)-1-oxy-nicotinamide |...)
Affinity DataIC50: >2.00E+4nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102214(6-Chloro-N-(4-fluoro-benzyl)-1-oxy-nicotinamide | ...)
Affinity DataIC50: >2.00E+4nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50102215(6-Chloro-N-(2-hydroxy-phenyl)-1-oxy-nicotinamide |...)
Affinity DataIC50: >2.00E+4nMAssay Description:Evaluated using an SPA assay with recombinant human [125I]-IL-8 and membranes preparedfrom Sf9 cells expressing human CXCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed