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Found 32 Enz. Inhib. hit(s) with all data for entry = 50011181
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103281(1-(3-Benzoyl-4-diphenylacetylamino-phenylcarbamoyl...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103269(1-{3-Benzoyl-4-[2-(4-bromo-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  76nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103285(1-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  77nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103271(1-(3-Benzoyl-4-phenylmethanesulfonylamino-phenylca...)
Affinity DataIC50:  85nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103280(1-(3-Benzoyl-4-p-tolylmethanesulfonylamino-phenylc...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103262(1-{3-Benzoyl-4-[2-(4-chloro-phenyl)-acetylamino]-p...)
Affinity DataIC50:  105nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103274(1-{3-Benzoyl-4-[2-(4-nitro-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  115nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103261(1-{3-Benzoyl-4-[2-(2,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103270(1-{3-Benzoyl-4-[2-(2,6-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103272(1-[3-Benzoyl-4-(2-naphthalen-1-yl-acetylamino)-phe...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103260(1-[3-Benzoyl-4-(2-o-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103258(1-{3-Benzoyl-4-[2-(2,3-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  420nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103277(1-[3-Benzoyl-4-(2-naphthalen-2-yl-acetylamino)-phe...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103284(1-{3-Benzoyl-4-[2-(3,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103276(1-{3-Benzoyl-4-[2-(3,5-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  535nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103259(1-[3-Benzoyl-4-(2-m-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  540nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103268(1-{3-Benzoyl-4-[2-(4-methoxy-phenyl)-acetylamino]-...)
Affinity DataIC50:  545nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103257(1-[3-Benzoyl-4-(4-carboxy-butyrylamino)-phenylcarb...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103278(1-[3-Benzoyl-4-(2-phenyl-propionylamino)-phenylcar...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103287(1-(3-Benzoyl-4-phenylacetylamino-phenylcarbamoyl)-...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103266(1-[3-Benzoyl-4-(3-carboxy-propionylamino)-phenylca...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103283(1-{3-Benzoyl-4-[2-(4-trifluoromethyl-phenyl)-acety...)
Affinity DataIC50:  725nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103282(1-[3-Benzoyl-4-(3-phenyl-propionylamino)-phenylcar...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103256(1-[3-Benzoyl-4-(2-oxo-2-phenyl-acetylamino)-phenyl...)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103263(1-[3-Benzoyl-4-(3-methoxycarbonyl-propionylamino)-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103267(1-[3-Benzoyl-4-(2-biphenyl-4-yl-acetylamino)-pheny...)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103273(1-{3-Benzoyl-4-[2-(2,5-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103264(1-[3-Benzoyl-4-(4-methoxycarbonyl-butyrylamino)-ph...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103265(1-{3-Benzoyl-4-[(naphthalene-1-carbonyl)-amino]-ph...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103286(1-(3-Benzoyl-4-benzoylamino-phenylcarbamoyl)-2-mer...)
Affinity DataIC50:  4.78E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103275(1-(4-Acetylamino-3-benzoyl-phenylcarbamoyl)-2-merc...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103279(1-[3-Benzoyl-4-(3,5,5-trimethyl-hexanoylamino)-phe...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed