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Found 42 Enz. Inhib. hit(s) with all data for entry = 50035173
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50066523(2,2,4-Trimethyl-6-(3-nitro-phenyl)-1,2-dihydro-qui...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105572(1-Benzyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataKi:  30nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105564(6-(3-Chloro-phenyl)-3H-benzothiazol-2-one | CHEMBL...)
Affinity DataKi:  127nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105561(1-Benzyl-6-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataKi:  150nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105566(6-(3-Nitro-phenyl)-3H-benzothiazol-2-one | CHEMBL3...)
Affinity DataKi:  332nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105563(1-Benzyl-6-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataKi:  521nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105565(6-(3-Chloro-phenyl)-1-isopropyl-1,3-dihydro-benzoi...)
Affinity DataKi:  525nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105560(1-Isopropyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoim...)
Affinity DataKi:  525nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105562(1-Benzyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataKi:  714nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105559(1-Benzyl-5-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataKi:  3.13E+3nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105568(1-Methyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105567(1-Benzyl-5-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105572(1-Benzyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105561(1-Benzyl-6-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataIC50:  17nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105571(6-(3-Chloro-phenyl)-1-ethyl-1,3-dihydro-benzoimida...)
Affinity DataIC50:  29nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50066523(2,2,4-Trimethyl-6-(3-nitro-phenyl)-1,2-dihydro-qui...)
Affinity DataIC50:  41nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50066523(2,2,4-Trimethyl-6-(3-nitro-phenyl)-1,2-dihydro-qui...)
Affinity DataIC50:  42nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105562(1-Benzyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataIC50:  62nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105560(1-Isopropyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoim...)
Affinity DataIC50:  73nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105566(6-(3-Nitro-phenyl)-3H-benzothiazol-2-one | CHEMBL3...)
Affinity DataIC50:  84nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105571(6-(3-Chloro-phenyl)-1-ethyl-1,3-dihydro-benzoimida...)
Affinity DataIC50:  106nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105565(6-(3-Chloro-phenyl)-1-isopropyl-1,3-dihydro-benzoi...)
Affinity DataIC50:  113nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105563(1-Benzyl-6-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataIC50:  113nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105560(1-Isopropyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoim...)
Affinity DataIC50:  136nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105562(1-Benzyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataIC50:  257nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105564(6-(3-Chloro-phenyl)-3H-benzothiazol-2-one | CHEMBL...)
Affinity DataIC50:  265nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105566(6-(3-Nitro-phenyl)-3H-benzothiazol-2-one | CHEMBL3...)
Affinity DataIC50:  326nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105565(6-(3-Chloro-phenyl)-1-isopropyl-1,3-dihydro-benzoi...)
Affinity DataIC50:  412nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105563(1-Benzyl-6-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataIC50:  412nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105564(6-(3-Chloro-phenyl)-3H-benzothiazol-2-one | CHEMBL...)
Affinity DataIC50:  460nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105570(6-(3-Chloro-phenyl)-1-methyl-1,3-dihydro-benzoimid...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105568(1-Methyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105570(6-(3-Chloro-phenyl)-1-methyl-1,3-dihydro-benzoimid...)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105568(1-Methyl-6-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105559(1-Benzyl-5-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibitory concentration against progesterone induced PRE-luciferase activity in CV-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105567(1-Benzyl-5-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105567(1-Benzyl-5-(3-nitro-phenyl)-1,3-dihydro-benzoimida...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards progesterone receptor was measuredMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105559(1-Benzyl-5-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50105569(1-Benzyl-5-(3-chloro-phenyl)-1,3-dihydro-benzoimid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration against progesterone stimulated alkaline phosphatase activity in T47D human breast carcinoma cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed