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Found 4 Enz. Inhib. hit(s) with all data for entry = 50011354
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of DNA-dependent protein kinase (DNA-PK) of HeLa cell nuclear cell extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50105673(2-Hydrazonomethyl-6-oxo-1,6-dihydro-[3,4']bipyridi...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of DNA-dependent protein kinase (DNA-PK) of HeLa cell nuclear cell extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50105672(CHEMBL329643 | Trifluoro-acetate5-cyano-2-hydroxym...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of DNA-dependent protein kinase (DNA-PK) of HeLa cell nuclear cell extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50105674(2-(4-Methoxy-benzyloxymethyl)-6-oxo-1,6-dihydro-[3...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of DNA-dependent protein kinase (DNA-PK) of HeLa cell nuclear cell extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed