Compile Data Set for Download or QSAR
maximum 50k data
Found 65 Enz. Inhib. hit(s) with all data for entry = 50011394
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106064((S)-2-(3-Carbamimidoyl-benzoyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106056((R)-2-(3-Carbamimidoyl-benzoyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106058(3-Carbamimidoyl-N-[(R)-2-phenyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106057(3-Carbamimidoyl-N-[(R)-phenyl-(2'-sulfamoyl-biphen...)
Affinity DataIC50:  35nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106059(3-Carbamimidoyl-N-[(R)-2-methyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50:  35nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106055((S)-3-(3-Carbamimidoyl-benzoylamino)-N-(2'-sulfamo...)
Affinity DataIC50:  55nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106051((S)-2-(3-Carbamimidoyl-benzoyl)-6-hydroxy-1,2,3,4-...)
Affinity DataIC50:  97nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106052(3-Carbamimidoyl-N-[(S)-phenyl-(2'-sulfamoyl-biphen...)
Affinity DataIC50:  337nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106063(3-Carbamimidoyl-N-[(S)-cyclohexyl-(2'-sulfamoyl-bi...)
Affinity DataIC50:  635nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106062((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50:  644nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106060(3-Carbamimidoyl-N-[(S)-2-methyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50:  676nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106050(3-Carbamimidoyl-N-[(S)-2-phenyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50:  762nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106053((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50:  842nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106069(3-Carbamimidoyl-N-[(2'-sulfamoyl-biphenyl-4-ylcarb...)
Affinity DataIC50:  851nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106051((S)-2-(3-Carbamimidoyl-benzoyl)-6-hydroxy-1,2,3,4-...)
Affinity DataIC50:  888nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106067((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50:  1.44E+3nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106057(3-Carbamimidoyl-N-[(R)-phenyl-(2'-sulfamoyl-biphen...)
Affinity DataIC50:  1.77E+3nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106049((R)-2-(3-Carbamimidoyl-benzoyl)-6-hydroxy-1,2,3,4-...)
Affinity DataIC50:  1.78E+3nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106064((S)-2-(3-Carbamimidoyl-benzoyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50:  2.15E+3nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106068((S)-2-(1-Amino-isoquinoline-7-carbonyl)-1,2,3,4-te...)
Affinity DataIC50:  2.77E+3nMAssay Description:Inhibitory activity of the compound against Coagulation factor X was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106066(3-Amino-1H-indazole-5-carboxylic acid [(R)-phenyl-...)
Affinity DataIC50:  3.45E+3nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106056((R)-2-(3-Carbamimidoyl-benzoyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50:  4.39E+3nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106055((S)-3-(3-Carbamimidoyl-benzoylamino)-N-(2'-sulfamo...)
Affinity DataIC50:  4.81E+3nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106052(3-Carbamimidoyl-N-[(S)-phenyl-(2'-sulfamoyl-biphen...)
Affinity DataIC50:  5.17E+3nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106062((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50:  5.64E+3nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106057(3-Carbamimidoyl-N-[(R)-phenyl-(2'-sulfamoyl-biphen...)
Affinity DataIC50:  6.56E+3nMAssay Description:Inhibitory activity of the compound against activated protein C (APC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106063(3-Carbamimidoyl-N-[(S)-cyclohexyl-(2'-sulfamoyl-bi...)
Affinity DataIC50: >7.93E+3nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106050(3-Carbamimidoyl-N-[(S)-2-phenyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106052(3-Carbamimidoyl-N-[(S)-phenyl-(2'-sulfamoyl-biphen...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106053((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106054(3-Amino-benzo[d]isoxazole-5-carboxylic acid [(R)-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106055((S)-3-(3-Carbamimidoyl-benzoylamino)-N-(2'-sulfamo...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106056((R)-2-(3-Carbamimidoyl-benzoyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106058(3-Carbamimidoyl-N-[(R)-2-phenyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106049((R)-2-(3-Carbamimidoyl-benzoyl)-6-hydroxy-1,2,3,4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106059(3-Carbamimidoyl-N-[(R)-2-methyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106060(3-Carbamimidoyl-N-[(S)-2-methyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106060(3-Carbamimidoyl-N-[(S)-2-methyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106061((S)-1-(3-Carbamimidoyl-benzoyl)-pyrrolidine-2-carb...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106061((S)-1-(3-Carbamimidoyl-benzoyl)-pyrrolidine-2-carb...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106058(3-Carbamimidoyl-N-[(R)-2-phenyl-1-(2'-sulfamoyl-bi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106054(3-Amino-benzo[d]isoxazole-5-carboxylic acid [(R)-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity of the compound against Coagulation factor X was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106065(3-Amino-1H-indazole-5-carboxylic acid [(S)-phenyl-...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106067((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106067((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106066(3-Amino-1H-indazole-5-carboxylic acid [(R)-phenyl-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106053((S)-4-(3-Carbamimidoyl-benzoylamino)-4-(2'-sulfamo...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106063(3-Carbamimidoyl-N-[(S)-cyclohexyl-(2'-sulfamoyl-bi...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106064((S)-2-(3-Carbamimidoyl-benzoyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Cor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50106069(3-Carbamimidoyl-N-[(2'-sulfamoyl-biphenyl-4-ylcarb...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 65 total ) | Next | Last >>
Jump to: