Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50011395
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM19807(CHEMBL100563 | benzyl N-[(1S)-1-({1-[(2S)-2-{[(ben...)
Affinity DataKi:  2nMAssay Description:Inhibitory activity of the compound against Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106075((S)-1-[2-Oxo-2-(3,4,5-trimethoxy-phenyl)-ethyl]-pi...)
Affinity DataKi:  790nMAssay Description:Inhibitory activity of the compound against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106079((S)-1-(2-Oxo-2-phenyl-ethyl)-piperidine-2-carboxyl...)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106077((S)-1-[2-(4-Chloro-phenyl)-2-oxo-ethyl]-piperidine...)
Affinity DataIC50:  280nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106076((S)-1-[2-(4-Methoxy-phenyl)-2-oxo-ethyl]-piperidin...)
Affinity DataIC50:  410nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106074((S)-1-(2-Oxo-2-phenyl-ethyl)-piperidine-2-carboxyl...)
Affinity DataIC50:  590nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106070((S)-1-(2-Benzo[1,3]dioxol-5-yl-2-oxo-ethyl)-piperi...)
Affinity DataIC50:  590nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106072((S)-1-[2-(2,6-Dimethoxy-phenyl)-2-oxo-ethyl]-piper...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106080((S)-1-(2-Oxo-2-phenyl-ethyl)-piperidine-2-carboxyl...)
Affinity DataIC50:  740nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106078((S)-1-(2-Oxo-2-phenyl-ethyl)-piperidine-2-carboxyl...)
Affinity DataIC50:  780nMAssay Description:Inhibitory activity of the compound against Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106081((S)-1-(2-Oxo-2-phenyl-ethyl)-piperidine-2-carboxyl...)
Affinity DataIC50:  840nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106075((S)-1-[2-Oxo-2-(3,4,5-trimethoxy-phenyl)-ethyl]-pi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106071((S)-1-(2-Oxo-2-phenyl-ethyl)-piperidine-2-carboxyl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50106073((S)-1-[2-Oxo-2-(3,4,5-trimethoxy-phenyl)-ethyl]-pi...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed