Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50011398
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106110(CHEMBL98692 | [1-(3-Methyl-3H-imidazol-4-ylmethyl)...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106112(CHEMBL101889 | [1-(3H-Imidazol-4-ylmethyl)-4-napht...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106113((4-Bromo-phenyl)-[1-(3H-imidazol-4-ylmethyl)-4-nap...)
Affinity DataIC50:  32nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106111(CHEMBL98806 | [1-(3H-Imidazol-4-ylmethyl)-4-naphth...)
Affinity DataIC50:  65nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106114((2-Bromo-phenyl)-[1-(3H-imidazol-4-ylmethyl)-4-nap...)
Affinity DataIC50:  88nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106117(CHEMBL102187 | [1-(3H-Imidazol-4-ylmethyl)-4-napht...)
Affinity DataIC50:  115nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106116((3-Bromo-phenyl)-[1-(3H-imidazol-4-ylmethyl)-4-nap...)
Affinity DataIC50:  150nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106118(CHEMBL319294 | [4-Anthracen-9-yl-1-(3H-imidazol-4-...)
Affinity DataIC50:  470nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106120(CHEMBL98498 | [1-(3H-Imidazol-4-ylmethyl)-4-naphth...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106119(CHEMBL101551 | [1-(3H-Imidazol-4-ylmethyl)-4-napht...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50106115(CHEMBL101897 | [1-(3H-Imidazol-4-ylmethyl)-4-pheny...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed