Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50011671
TargetInterstitial collagenase(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109171(CHEMBL122591 | [(S)-1-((S)-1-Methyl-2-oxo-ethylcar...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109168((R)-N*1*-[(S)-1-((S)-1-Formyl-3-methyl-butylcarbam...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109167((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-(2-oxo-eth...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109169((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-((S)-1-met...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109170(CHEMBL125553 | N*4*-Hydroxy-2-isobutyl-N*1*-[3-met...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109169((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-((S)-1-met...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109172((R)-N*1*-[(S)-1-((S)-2,2-Diethoxy-1-methyl-ethylca...)
Affinity DataIC50:  29nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109170(CHEMBL125553 | N*4*-Hydroxy-2-isobutyl-N*1*-[3-met...)
Affinity DataIC50:  47nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50031795((N-(2-HYDROXAMATEMETHYLENE-4-METHYL-PENTOYL)PHENYL...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109171(CHEMBL122591 | [(S)-1-((S)-1-Methyl-2-oxo-ethylcar...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109172((R)-N*1*-[(S)-1-((S)-2,2-Diethoxy-1-methyl-ethylca...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109168((R)-N*1*-[(S)-1-((S)-1-Formyl-3-methyl-butylcarbam...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50109167((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-(2-oxo-eth...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of Cathepsin L from human kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed