Compile Data Set for Download or QSAR
maximum 50k data
Found 53 Enz. Inhib. hit(s) with all data for entry = 50035236
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  3.10nMAssay Description:Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  5.90nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataKi:  12nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  16nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  18nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  21nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  28nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  28nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115718(1-Phenyl-4-(4-phenylethynyl-1H-pyrrol-2-ylmethyl)-...)
Affinity DataKi:  83nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115719(1-Phenyl-4-(1H-pyrrol-2-ylmethyl)-piperazine | CHE...)
Affinity DataKi:  100nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataKi:  170nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataKi:  230nMAssay Description:Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  270nMAssay Description:Ability to displace [3H]8-OH-DPAT radioligand from porcine 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  380nMAssay Description:Ability to displace [3H]-Ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  420nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  450nMAssay Description:Ability to displace [3H]8-OH-DPAT radioligand from porcine 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  510nMAssay Description:Ability to displace [3H]8-OH-DPAT radioligand from porcine 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataKi:  540nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115718(1-Phenyl-4-(4-phenylethynyl-1H-pyrrol-2-ylmethyl)-...)
Affinity DataKi:  550nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115719(1-Phenyl-4-(1H-pyrrol-2-ylmethyl)-piperazine | CHE...)
Affinity DataKi:  570nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  580nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  610nMAssay Description:Ability to displace [3H]-Ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115718(1-Phenyl-4-(4-phenylethynyl-1H-pyrrol-2-ylmethyl)-...)
Affinity DataKi:  670nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  720nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115718(1-Phenyl-4-(4-phenylethynyl-1H-pyrrol-2-ylmethyl)-...)
Affinity DataKi:  760nMAssay Description:Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  770nMAssay Description:Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataKi:  790nMAssay Description:Ability to displace [3H]8-OH-DPAT radioligand from porcine 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  850nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  850nMAssay Description:Ability to displace [3H]-Ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  960nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  1.20E+3nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataKi:  1.30E+3nMAssay Description:Ability to displace [3H]-Ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  1.80E+3nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  2.00E+3nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataKi:  2.10E+3nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  2.40E+3nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115718(1-Phenyl-4-(4-phenylethynyl-1H-pyrrol-2-ylmethyl)-...)
Affinity DataKi:  2.70E+3nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115719(1-Phenyl-4-(1H-pyrrol-2-ylmethyl)-piperazine | CHE...)
Affinity DataKi:  3.00E+3nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115719(1-Phenyl-4-(1H-pyrrol-2-ylmethyl)-piperazine | CHE...)
Affinity DataKi:  3.10E+3nMAssay Description:Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  3.40E+3nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  3.70E+3nMAssay Description:Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  4.30E+3nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  4.30E+3nMAssay Description:Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  4.60E+3nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  5.00E+3nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115719(1-Phenyl-4-(1H-pyrrol-2-ylmethyl)-piperazine | CHE...)
Affinity DataKi:  5.40E+3nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  8.00E+3nMAssay Description:Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50073805(3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyra...)
Affinity DataKi:  1.20E+4nMAssay Description:Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115716(1-Phenyl-4-(4-phenyl-1H-pyrrol-2-ylmethyl)-piperaz...)
Affinity DataEC50:  6.80nMAssay Description:Effective concentration of compound required against human Dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataEC50:  1.90nMAssay Description:Effective concentration of compound required against human Dopamine D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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