Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50012616
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  10nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  12nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  16nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  16nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  18nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  20nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  25nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121048(2-[3-Butyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  28nMAssay Description:Binding affinity of second enantiomer (E2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  30nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  40nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  110nMAssay Description:Binding affinity of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50:  190nMAssay Description:Binding affinity of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  190nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity of first enantiomer (E1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121048(2-[3-Butyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121047(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121046(2-[3-(1-Hydroxy-ethyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121045(2-[3-Ethyl-5-(1-hydroxy-ethyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity of first diastereomer (D1) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109322(CHEMBL114761 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  7.00E+3nMAssay Description:Binding affinity of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50121049(5-Fluoro-2-[3-(1-hydroxy-ethyl)-2,6-diisopropyl-5-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Binding affinity of second diastereomer (D2) of the compound against human glucagon receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed