Compile Data Set for Download or QSAR
maximum 50k data
Found 43 Enz. Inhib. hit(s) with all data for entry = 50037237
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125842(5-amino(imino)methylamino-2-[1-[2-amino-3-phenyl-(...)
Affinity DataIC50:  0.00170nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM29388(Exanta | Melagatran | US11584714, Compound 999)
Affinity DataIC50:  4.70nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125849(CHEMBL17587 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  49nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125847(CHEMBL275154 | Cyclopent-2-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  73nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125851(CHEMBL17455 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  210nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125837(CHEMBL17311 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125853(CHEMBL17139 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  240nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125870(CHEMBL17636 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125864(CHEMBL17365 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125848(CHEMBL17024 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  270nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125852(CHEMBL17465 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125840(CHEMBL418728 | Cyclopent-2-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  390nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125856(CHEMBL17508 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  630nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125862(CHEMBL273810 | Cyclopent-2-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  680nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125861(CHEMBL17464 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  940nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125838(CHEMBL416905 | Cyclopent-2-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  970nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125859(CHEMBL17745 | {[5-(4-Carbamimidoyl-benzylcarbamoyl...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50087830(CHEMBL49808 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50370293(CHEMBL1907917)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125863(2-(2-Methyl-2,3-dihydro-indole-1-carbonyl)-cyclope...)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125860(CHEMBL17253 | Cyclohex-2-ene-1,2-dicarboxylic acid...)
Affinity DataIC50:  3.80E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125855(CHEMBL17381 | Cyclohex-2-ene-1,2-dicarboxylic acid...)
Affinity DataIC50:  4.60E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125841(2-(2,3-Dihydro-indole-1-carbonyl)-cyclopent-2-enec...)
Affinity DataIC50:  4.60E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125869(CHEMBL416904 | Cyclopent-2-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  4.90E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125874(2-(Piperidine-1-carbonyl)-cyclopent-2-enecarboxyli...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125843(CHEMBL17553 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  7.80E+3nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125871(CHEMBL17646 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  1.12E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125845(CHEMBL279594 | Cyclopent-2-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  1.60E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125868(CHEMBL17786 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  1.90E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125867(CHEMBL17225 | Cyclopent-1-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  1.90E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125873(5-(2,3-Dihydro-indole-1-carbonyl)-cyclopent-1-enec...)
Affinity DataIC50:  2.20E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125857(CHEMBL274021 | Cyclopent-1-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125866(CHEMBL418729 | Cyclopent-1-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  2.40E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125835(CHEMBL273591 | Cyclopent-1-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  2.80E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125865(CHEMBL265586 | Cyclopent-1-ene-1,2-dicarboxylic ac...)
Affinity DataIC50:  3.30E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125846(2-(Piperidine-1-carbonyl)-cyclohex-2-enecarboxylic...)
Affinity DataIC50:  3.80E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125836(CHEMBL17781 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  5.80E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125834(CHEMBL17712 | Cyclopent-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50:  9.30E+4nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125854(CHEMBL17475 | Cyclohex-2-ene-1,2-dicarboxylic acid...)
Affinity DataIC50:  1.09E+5nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125875(CHEMBL17068 | {[2-(4-Carbamimidoyl-benzylcarbamoyl...)
Affinity DataIC50:  1.20E+5nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125844(CHEMBL17515 | Cyclohex-2-ene-1,2-dicarboxylic acid...)
Affinity DataIC50:  1.30E+5nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125872(2-(2,3-Dihydro-indole-1-carbonyl)-cyclopent-1-enec...)
Affinity DataIC50: >1.30E+5nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Link£Ping University

Curated by ChEMBL
LigandPNGBDBM50125850(CHEMBL278282 | Cyclohex-2-ene-1,2-dicarboxylic aci...)
Affinity DataIC50: >1.30E+5nMAssay Description:In vitro inhibitory concentration of compound against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed