Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50013428
TargetMetabotropic glutamate receptor 1(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 1 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM50130516((+/-)-(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-...)
Affinity DataKi:  9.40E+4nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 1 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Affinity DataKi:  4.40E+5nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 5 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50130516((+/-)-(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-...)
Affinity DataKi:  6.40E+5nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 5 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50130516((+/-)-(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 4 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 4 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM66976((1S,3R)-1-aminocyclopentane-1,3-dicarboxylic acid;...)
Affinity DataEC50:  2.00E+3nMAssay Description:Activity of the compound tested at cloned rat mGluR2 receptor expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM66976((1S,3R)-1-aminocyclopentane-1,3-dicarboxylic acid;...)
Affinity DataEC50:  2.30E+4nMAssay Description:Activity of the compound tested at cloned rat Metabotropic glutamate receptor 5 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Affinity DataEC50: >1.00E+6nMAssay Description:Activity of the compound tested at cloned rat Metabotropic glutamate receptor 4 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM66976((1S,3R)-1-aminocyclopentane-1,3-dicarboxylic acid;...)
Affinity DataEC50:  8.00E+5nMAssay Description:Activity of the compound tested at cloned rat Metabotropic glutamate receptor 4 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50130516((+/-)-(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-...)
Affinity DataEC50: >1.00E+6nMAssay Description:Activity of the compound tested at cloned rat Metabotropic glutamate receptor 4 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Affinity DataEC50:  1.60E+4nMAssay Description:Activity of the compound tested at cloned rat mGluR2 receptor expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Università

Curated by ChEMBL
LigandPNGBDBM66976((1S,3R)-1-aminocyclopentane-1,3-dicarboxylic acid;...)
Affinity DataEC50:  1.50E+4nMAssay Description:Activity of the compound tested at cloned rat Metabotropic glutamate receptor 1 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed