Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50000055
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataKi:  98nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000717(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...)
Affinity DataKi:  142nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000701(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...)
Affinity DataKi:  157nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000707(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...)
Affinity DataKi:  167nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000722(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...)
Affinity DataKi:  331nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000720(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...)
Affinity DataKi:  345nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000719(CHEMBL62812 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...)
Affinity DataKi:  390nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000708(4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...)
Affinity DataKi:  656nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000700(4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...)
Affinity DataKi:  690nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000716(CHEMBL61680 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...)
Affinity DataKi:  925nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000718(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...)
Affinity DataKi:  945nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000705(2-({7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydro...)
Affinity DataKi:  1.58E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000712(7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-dimet...)
Affinity DataKi:  3.25E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000711(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...)
Affinity DataKi:  3.30E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000715(2-[7-(1,2-Dimethyl-heptyl)-5-hydroxy-10,10-dimethy...)
Affinity DataKi:  3.68E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000702(7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methoxy-1...)
Affinity DataKi:  4.21E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000710(3-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...)
Affinity DataKi:  4.40E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000699(3-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...)
Affinity DataKi:  5.50E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000709(5-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...)
Affinity DataKi:  5.50E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000724(2-(5-Hydroxy-7-isopropyl-10,10-dimethyl-1,2,4,10-t...)
Affinity DataKi:  9.00E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000725(7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-dimet...)
Affinity DataKi:  1.18E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000721(2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...)
Affinity DataKi:  1.58E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000703(7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methoxy-1...)
Affinity DataKi:  1.69E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000723(1-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...)
Affinity DataKi:  2.05E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000726(4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...)
Affinity DataKi:  2.07E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000713(2-[5-{4-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-2,6-d...)
Affinity DataKi:  2.35E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000706(6-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...)
Affinity DataKi:  2.50E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50000704(7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-1,4,4-trime...)
Affinity DataKi:  4.38E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed