Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50000260
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003669(Ac-Tyr(SO3H)-Met-Gly-Trp-Met-R-Dtc-Phe-NH2 | CHEMB...)
Affinity DataIC50:  0.0500nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003666(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003670(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  0.600nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003667(4-{2-Acetylamino-2-[1-({[1-{1-[2-carbamoyl-1-(1-ca...)
Affinity DataIC50:  1.40nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003664(4-{2-Acetylamino-2-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataIC50:  2.40nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003670(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  4.40nMAssay Description:Concentration of the compound inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003665(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  5.5nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003662(4-{2-Acetylamino-2-[1-({[1-{1-[2-(1-carbamoyl-2-ph...)
Affinity DataIC50:  8.30nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003665(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  22nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003668(CHEMBL3143146 | [1-[1-[4-(1-Carbamoyl-2-phenyl-eth...)
Affinity DataIC50:  59nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003664(4-{2-Acetylamino-2-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataIC50:  170nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003667(4-{2-Acetylamino-2-[1-({[1-{1-[2-carbamoyl-1-(1-ca...)
Affinity DataIC50:  200nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003663(Ac-Tyr(SO3H)-Met-Gly-Trp-Met-S-Dtc-Phe-NH2 | CHEMB...)
Affinity DataIC50:  314nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003666(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from bovine striatal binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003669(Ac-Tyr(SO3H)-Met-Gly-Trp-Met-R-Dtc-Phe-NH2 | CHEMB...)
Affinity DataIC50:  2.31E+3nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003662(4-{2-Acetylamino-2-[1-({[1-{1-[2-(1-carbamoyl-2-ph...)
Affinity DataIC50:  3.90E+3nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003663(Ac-Tyr(SO3H)-Met-Gly-Trp-Met-S-Dtc-Phe-NH2 | CHEMB...)
Affinity DataIC50:  6.16E+3nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003668(CHEMBL3143146 | [1-[1-[4-(1-Carbamoyl-2-phenyl-eth...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from bovine striatal binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed