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Found 17 Enz. Inhib. hit(s) with all data for entry = 50014022
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137236(5-Acetylamino-2-{[2-(3-fluoro-4-trifluoromethyl-ph...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137238(2-{[2-(3-Fluoro-4-trifluoromethyl-phenyl)-5-oxo-ox...)
Affinity DataIC50:  270nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137242(5-Methyl-2-{[5-oxo-2-(4-trifluoromethyl-phenyl)-ox...)
Affinity DataIC50:  830nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137227(5-Chloro-2-{[2-(3-fluoro-4-trifluoromethyl-phenyl)...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137229(2-{[2-(4-Chloro-phenyl)-5-oxo-oxazol-(4E)-ylidenem...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137234(5-Bromo-2-{[2-(3-fluoro-4-trifluoromethyl-phenyl)-...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137233(5-Fluoro-2-{[5-oxo-2-(4-trifluoromethyl-phenyl)-ox...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137235(5-Bromo-4-chloro-2-{[5-oxo-2-(4-trifluoromethyl-ph...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137239(2-{[2-(4-Chloro-phenyl)-5-oxo-oxazol-(4E)-ylidenem...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137230(5-Bromo-2-{[2-(4-chloro-phenyl)-5-oxo-oxazol-(4E)-...)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137231(5-Methyl-2-{[5-oxo-2-(3-trifluoromethoxy-phenyl)-o...)
Affinity DataIC50:  4.40E+3nMAssay Description:In vitro inhibitory activity against acyl carrier protein synthase (AcpS) in Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137237(5-Bromo-2-{[5-oxo-2-(3-trifluoromethoxy-phenyl)-ox...)
Affinity DataIC50:  1.50E+4nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137240(2-{[2-(4-Chloro-phenyl)-5-oxo-oxazol-(4E)-ylidenem...)
Affinity DataIC50:  1.50E+4nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137243(2-{[5-Oxo-2-phenyl-oxazol-(4E)-ylidenemethyl]-amin...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137241(5-Bromo-4-chloro-2-{[2-(4-chloro-phenyl)-5-oxo-oxa...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137232(5-Chloro-2-{[5-oxo-2-(3-trifluoromethoxy-phenyl)-o...)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHolo-[acyl-carrier-protein] synthase(Bacillus subtilis)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50137228(5-Fluoro-2-{[2-(4-methoxy-phenyl)-5-oxo-oxazol-(4E...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against Holo-[acyl-carrier-protein] synthase was determined using Bacillus subtilis GST-Acp-HTRFassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed