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Found 24 Enz. Inhib. hit(s) with all data for entry = 50035445
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221787(CHEMBL3216418)
Affinity DataKi:  0.0420nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221778(CHEMBL3216392)
Affinity DataKi:  0.114nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221781(CHEMBL3215968)
Affinity DataKi:  0.115nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221780(CHEMBL3217089)
Affinity DataKi:  1.20nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221781(CHEMBL3215968)
Affinity DataKi:  7.30nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221787(CHEMBL3216418)
Affinity DataKi:  13nMAssay Description:pA2 is the negative log of the molar concentration required to double the agonism of opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221780(CHEMBL3217089)
Affinity DataKi:  16nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221778(CHEMBL3216392)
Affinity DataKi:  23nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221779(CHEMBL3215974)
Affinity DataKi:  26nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221782(CHEMBL3215530)
Affinity DataKi:  70nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146023(2-Amino-N-[2-(5-{2-[2-amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  309nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221779(CHEMBL3215974)
Affinity DataKi:  435nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146020(2-Amino-N-(5-{[2-amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  460nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146020(2-Amino-N-(5-{[2-amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  1.83E+3nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221782(CHEMBL3215530)
Affinity DataKi:  2.19E+3nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50146023(2-Amino-N-[2-(5-{2-[2-amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  2.90E+3nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221787(CHEMBL3216418)
Affinity DataIC50:  1.30nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221778(CHEMBL3216392)
Affinity DataIC50:  1.90nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221781(CHEMBL3215968)
Affinity DataIC50:  13nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221778(CHEMBL3216392)
Affinity DataIC50:  42nMAssay Description:pA2 is the negative log of the molar concentration required to double the agonism of opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221787(CHEMBL3216418)
Affinity DataIC50: >1.00E+3nMAssay Description:Compound was tested for opioid receptor delta 1 agonism or antagonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221780(CHEMBL3217089)
Affinity DataIC50:  1.70E+3nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221781(CHEMBL3215968)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for opioid receptor delta 1 agonism or antagonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institutes Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50221780(CHEMBL3217089)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed