Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50037329
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152761(3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-b...)
Affinity DataIC50:  7nMAssay Description:Concentration required to inhibit [125I]IL-8 binding towards C-X-C chemokine receptor type 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152759(3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-b...)
Affinity DataIC50:  10nMAssay Description:Concentration required to inhibit [125I]IL-8 binding towards C-X-C chemokine receptor type 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152760(3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-N...)
Affinity DataIC50:  12nMAssay Description:Concentration required to inhibit [125I]IL-8 binding towards C-X-C chemokine receptor type 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152762(1-(2-Bromo-phenyl)-3-(3,4-dichloro-2-hydroxy-pheny...)
Affinity DataIC50:  63nMAssay Description:Concentration required to inhibit [125I]IL-8 binding towards C-X-C chemokine receptor type 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152763(1-(3-Aminomethyl-4-chloro-2-hydroxy-phenyl)-3-(2-b...)
Affinity DataIC50:  114nMAssay Description:Concentration required to inhibit [125I]IL-8 binding towards C-X-C chemokine receptor type 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152764(1-(2-Bromo-phenyl)-3-(4-chloro-2-hydroxy-phenyl)-u...)
Affinity DataIC50:  906nMAssay Description:Concentration required to inhibit [125I]IL-8 binding towards C-X-C chemokine receptor type 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152761(3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-b...)
Affinity DataIC50:  1.37E+3nMAssay Description:Concentration required to inhibit [125I]-IL-8 binding towards C-X-C chemokine receptor type 1 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152760(3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-N...)
Affinity DataIC50:  4.32E+3nMAssay Description:Concentration required to inhibit [125I]-IL-8 binding towards C-X-C chemokine receptor type 1 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152759(3-[3-(2-Bromo-phenyl)-ureido]-6-chloro-2-hydroxy-b...)
Affinity DataIC50:  6.04E+3nMAssay Description:Concentration required to inhibit [125I]-IL-8 binding towards C-X-C chemokine receptor type 1 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152762(1-(2-Bromo-phenyl)-3-(3,4-dichloro-2-hydroxy-pheny...)
Affinity DataIC50:  1.34E+4nMAssay Description:Concentration required to inhibit [125I]-IL-8 binding towards C-X-C chemokine receptor type 1 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50152763(1-(3-Aminomethyl-4-chloro-2-hydroxy-phenyl)-3-(2-b...)
Affinity DataIC50:  3.00E+4nMAssay Description:Concentration required to inhibit [125I]-IL-8 binding towards C-X-C chemokine receptor type 1 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed