TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 108nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 108nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 201nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 201nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 217nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 223nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 229nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 247nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 271nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 287nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 288nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 307nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 309nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 312nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 318nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 334nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 335nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 337nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 342nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 359nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 376nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 389nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 418nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 418nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 445nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 451nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 451nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 461nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 497nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 575nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 664nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 806nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 824nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 875nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 882nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 949nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 966nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 982nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair