Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50000412
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005459(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Affinity DataKi:  49nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005456(1-(4-Chloro-phenyl)-3-(3,3-diphenyl-allyl)-urea | ...)
Affinity DataKi:  90nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005471(1H-Indole-2-carboxylic acid (3-phenyl-allyl)-amide...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005453(1H-Indole-2-carboxylic acid [3,3-bis-(4-chloro-phe...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005450(1-(4-Chloro-phenyl)-3-(3-pentyl-oct-2-enyl)-urea |...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005455(1H-Indole-2-carboxylic acid (3,3-diphenyl-propyl)-...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005466(1H-Indole-2-carboxylic acid (3,3-diphenyl-allyl)-a...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005468(3,4-Dichloro-N-(3,3-diphenyl-allyl)-benzamide | CH...)
Affinity DataKi:  400nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005457(1-(4-Chloro-phenyl)-3-(4,4-diphenyl-but-3-enyl)-ur...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005470(CHEMBL8949 | Naphthalene-2-carboxylic acid (3,3-di...)
Affinity DataKi:  450nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005461(CHEMBL9510 | Quinoline-2-carboxylic acid (3,3-diph...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005469(1-(3,3-Diphenyl-allyl)-3-m-tolyl-urea | CHEMBL9312)
Affinity DataKi:  800nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005462(CHEMBL9379 | Naphthalene-1-carboxylic acid (3,3-di...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005467(1-(4-Chloro-phenyl)-3-(2-diphenylamino-ethyl)-urea...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005465(4-Chloro-N-(3,3-diphenyl-allyl)-benzamide | CHEMBL...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005449(CHEMBL9174 | Quinoline-3-carboxylic acid (3,3-diph...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005460(5,6-Dihydro-4H-pyrrolo[3,2,1-ij]quinoline-2-carbox...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005452(1H-Indole-2-carboxylic acid (4,4-diphenyl-but-3-en...)
Affinity DataKi: >2.00E+3nMAssay Description:Compound was evaluated for its ability to inhibit [3H]-L-364,718 binding Cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005454(CHEMBL9181 | Quinoline-4-carboxylic acid (3,3-diph...)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005464(1-(4-Chloro-phenyl)-3-[2-(10,11-dihydro-dibenzo[a,...)
Affinity DataKi: >4.00E+3nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005458(1-(4-Chloro-phenyl)-3-(3-phenyl-allyl)-urea | CHEM...)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005451(1H-Indole-2-carboxylic acid [3,3-bis-(4-methoxy-ph...)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed