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Found 126 Enz. Inhib. hit(s) with all data for entry = 50015642
LigandPNGBDBM20464((2E)-3-[2-(piperidin-1-yl)-6-(trifluoromethyl)pyri...)
Affinity DataIC50:  0.420nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20464((2E)-3-[2-(piperidin-1-yl)-6-(trifluoromethyl)pyri...)
Affinity DataIC50:  1nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158665((E)-3-(4-tert-Butyl-phenyl)-N-quinolin-7-yl-acryla...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158658((E)-3-(2-Morpholin-4-yl-6-trifluoromethyl-pyridin-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158658((E)-3-(2-Morpholin-4-yl-6-trifluoromethyl-pyridin-...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158665((E)-3-(4-tert-Butyl-phenyl)-N-quinolin-7-yl-acryla...)
Affinity DataIC50:  2nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158681((E)-3-(4-tert-Butyl-phenyl)-N-(2-oxo-1,2,3,4-tetra...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158679((E)-3-(4-tert-Butyl-phenyl)-N-(3-oxo-3,4-dihydro-2...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158678((E)-3-(4-tert-Butyl-phenyl)-4-phenyl-but-2-enoic a...)
Affinity DataIC50:  14nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158647((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2-mor...)
Affinity DataIC50:  15nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158628(5-tert-Butyl-2-[(E)-2-(2,3-dihydro-benzo[1,4]dioxi...)
Affinity DataIC50:  15nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158633((E)-3-(4-tert-Butyl-phenyl)-5-methyl-hex-2-enoic a...)
Affinity DataIC50:  16nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158683((E)-3-(4-tert-Butyl-phenyl)-N-(3,4-dihydro-2H-benz...)
Affinity DataIC50:  16nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158634((E)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  20nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158671((E)-3-(4-tert-Butyl-phenyl)-N-(3-methoxy-phenyl)-a...)
Affinity DataIC50:  21nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158655((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  25nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158628(5-tert-Butyl-2-[(E)-2-(2,3-dihydro-benzo[1,4]dioxi...)
Affinity DataIC50:  26nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158649((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(6''-t...)
Affinity DataIC50:  27nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158640((E)-3-(4-tert-Butyl-phenyl)-N-(3-hydroxy-4-methoxy...)
Affinity DataIC50:  30nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158630((E)-3-(4-tert-Butyl-phenyl)-N-(1,2,3,4-tetrahydro-...)
Affinity DataIC50:  36nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158646((E)-4-(4-tert-Butyl-phenyl)-5-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  36nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158664((E)-3-(4-tert-Butyl-phenyl)-but-2-enoic acid (2,3-...)
Affinity DataIC50:  39nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158647((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2-mor...)
Affinity DataIC50:  40nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158632((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  44nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158666((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-tri...)
Affinity DataIC50:  46nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158649((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(6''-t...)
Affinity DataIC50:  54nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158668((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-iso...)
Affinity DataIC50:  55nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158683((E)-3-(4-tert-Butyl-phenyl)-N-(3,4-dihydro-2H-benz...)
Affinity DataIC50:  57nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158667((E)-3-(2-Bromo-4-tert-butyl-phenyl)-N-(2,3-dihydro...)
Affinity DataIC50:  60nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158643((E)-3-(4-tert-Butyl-phenyl)-N-(5,6,7,8-tetrahydro-...)
Affinity DataIC50:  61nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158681((E)-3-(4-tert-Butyl-phenyl)-N-(2-oxo-1,2,3,4-tetra...)
Affinity DataIC50:  71nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158650((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  78nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158668((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-iso...)
Affinity DataIC50:  82nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158633((E)-3-(4-tert-Butyl-phenyl)-5-methyl-hex-2-enoic a...)
Affinity DataIC50:  94nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158666((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-tri...)
Affinity DataIC50:  100nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158662((E)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  100nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158685((E)-3-(6-tert-Butyl-pyridin-3-yl)-N-(2,3-dihydro-b...)
Affinity DataIC50:  100nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158678((E)-3-(4-tert-Butyl-phenyl)-4-phenyl-but-2-enoic a...)
Affinity DataIC50:  110nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158682((E)-3-(4-tert-Butyl-phenyl)-N-(3,4-dihydro-2H-benz...)
Affinity DataIC50:  110nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158636((E)-3-(4-Bromo-phenyl)-N-(2,3-dihydro-benzo[1,4]di...)
Affinity DataIC50:  110nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158634((E)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  120nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158645((E)-3-(4-tert-Butyl-phenyl)-N-(4-methoxy-phenyl)-a...)
Affinity DataIC50:  140nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158644(3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1,4]d...)
Affinity DataIC50:  150nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158630((E)-3-(4-tert-Butyl-phenyl)-N-(1,2,3,4-tetrahydro-...)
Affinity DataIC50:  160nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158680((E)-3-(4-tert-Butyl-phenyl)-N-(3,4-dimethoxy-pheny...)
Affinity DataIC50:  170nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158629((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-eth...)
Affinity DataIC50:  170nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158655((Z)-3-(4-tert-Butyl-phenyl)-N-(2,3-dihydro-benzo[1...)
Affinity DataIC50:  180nMAssay Description:Inhibition of pH-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158676((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-nit...)
Affinity DataIC50:  190nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158674(2-(4-tert-butylbenzylidene)-N-(2,3-dihydrobenzo[b]...)
Affinity DataIC50:  210nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158670((E)-N-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-p-toly...)
Affinity DataIC50:  210nMAssay Description:Inhibition of capsaicin-induced calcium uptake by transient receptor potential vanilloid type 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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