Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 5495
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM82411(CAS_75921-69-6 | NDP-MSH)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86683(NBI-58702)
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM50152808((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  9.55nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86681(NBI-58704)
Affinity DataKi:  13.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86682(Beta MSH | CAS_114843 | NSC_114843)
Affinity DataKi:  18.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM86684(NBI-56297)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM82406(desacetyl-alpha-MSH)
Affinity DataKi:  30.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM50152798(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataKi:  74.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by PDSP Ki Database
LigandPNGBDBM82407(Gamma1-MSH)
Affinity DataKi:  589nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed