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Found 26 Enz. Inhib. hit(s) with all data for entry = 50016324
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM19441(2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethox...)
Affinity DataIC50:  0.890nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM19441(2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethox...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167734(10-[4-(2-Piperidin-1-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  2.84nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167736(10-[4-(2-Azepan-1-yl-ethoxy)-benzyl]-10H-benzo[4,5...)
Affinity DataIC50:  3.34nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167735(10-[4-(2-Pyrrolidin-1-yl-ethoxy)-benzyl]-10H-benzo...)
Affinity DataIC50:  6nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167736(10-[4-(2-Azepan-1-yl-ethoxy)-benzyl]-10H-benzo[4,5...)
Affinity DataIC50:  7.26nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167738(10-[4-(2-Morpholin-4-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  10nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167734(10-[4-(2-Piperidin-1-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167741(10-[4-(2-Diethylamino-ethoxy)-benzyl]-10H-benzo[4,...)
Affinity DataIC50:  16.4nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167732(10-[4-(2-Azepan-1-yl-ethoxy)-benzyl]-10H-benzo[4,5...)
Affinity DataIC50:  16.6nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167739(10-[4-(2-Dimethylamino-ethoxy)-benzyl]-10H-benzo[4...)
Affinity DataIC50:  18nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167732(10-[4-(2-Azepan-1-yl-ethoxy)-benzyl]-10H-benzo[4,5...)
Affinity DataIC50:  18nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167735(10-[4-(2-Pyrrolidin-1-yl-ethoxy)-benzyl]-10H-benzo...)
Affinity DataIC50:  20.2nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167738(10-[4-(2-Morpholin-4-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  21.4nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167737(10-[4-(2-Diethylamino-ethoxy)-benzyl]-10H-benzo[4,...)
Affinity DataIC50:  25nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167742(10-[4-(2-Pyrrolidin-1-yl-ethoxy)-benzyl]-10H-benzo...)
Affinity DataIC50:  27.2nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167739(10-[4-(2-Dimethylamino-ethoxy)-benzyl]-10H-benzo[4...)
Affinity DataIC50:  31nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167741(10-[4-(2-Diethylamino-ethoxy)-benzyl]-10H-benzo[4,...)
Affinity DataIC50:  31.2nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167733(10-[4-(2-Piperidin-1-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  35nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167733(10-[4-(2-Piperidin-1-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  39nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167740(10-[4-(2-Dimethylamino-ethoxy)-benzyl]-10H-benzo[4...)
Affinity DataIC50:  45.6nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167740(10-[4-(2-Dimethylamino-ethoxy)-benzyl]-10H-benzo[4...)
Affinity DataIC50:  51.4nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167742(10-[4-(2-Pyrrolidin-1-yl-ethoxy)-benzyl]-10H-benzo...)
Affinity DataIC50:  53.9nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167737(10-[4-(2-Diethylamino-ethoxy)-benzyl]-10H-benzo[4,...)
Affinity DataIC50:  57.4nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167731(10-[4-(2-Morpholin-4-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  126nMAssay Description:Inhibitino of [3H]-17-beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50167731(10-[4-(2-Morpholin-4-yl-ethoxy)-benzyl]-10H-benzo[...)
Affinity DataIC50:  215nMAssay Description:Inhibition of [3H]-17-beta-estradiol binding to human estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed