Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50016477
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169540(CHEMBL186479 | Cyclopropylmethyl-(2,2,2-trifluoro-...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169535(CHEMBL363592 | Dipropyl-[2-trifluoromethyl-9-(2,4,...)
Affinity DataKi:  11nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169517(CHEMBL190745 | Cyclopropylmethyl-[2-trifluoromethy...)
Affinity DataKi:  13nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169508(CHEMBL424812 | Cyclopropylmethyl-[2-methyl-9-(2,4,...)
Affinity DataKi:  20nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169531(CHEMBL188523 | Cyclopropylmethyl-[2-ethyl-9-(2,4,6...)
Affinity DataKi:  21nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169524(CHEMBL186628 | Cyclopropylmethyl-propyl-[2-trifluo...)
Affinity DataKi:  23nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169520(CHEMBL188813 | Cyclobutylmethyl-propyl-[2-trifluor...)
Affinity DataKi:  26nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169533(CHEMBL365715 | Cyclopropylmethyl-ethyl-[2-trifluor...)
Affinity DataKi:  28nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169523(CHEMBL427527 | Cyclopropylmethyl-(2,2,3,3,3-pentaf...)
Affinity DataKi:  34nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169498(CHEMBL191052 | Cyclobutylmethyl-(2,2,2-trifluoro-e...)
Affinity DataKi:  53nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169537(CHEMBL191366 | [9-(2-Bromo-4-isopropyl-phenyl)-2-t...)
Affinity DataKi:  54nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169529(CHEMBL360185 | Cyclopropylmethyl-[6-fluoro-2-methy...)
Affinity DataKi:  59nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169526(CHEMBL364002 | Propyl-[2-trifluoromethyl-9-(2,4,6-...)
Affinity DataKi:  68nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169511((2,2,3,3,3-Pentafluoro-propyl)-propyl-[2-trifluoro...)
Affinity DataKi:  75nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169515(CHEMBL189115 | Propyl-(2,2,2-trifluoro-ethyl)-[2-t...)
Affinity DataKi:  75nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169507(CHEMBL188194 | Diallyl-[2-trifluoromethyl-9-(2,4,6...)
Affinity DataKi:  138nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169509(CHEMBL187940 | Cyclopropylmethyl-[2-ethyl-6-fluoro...)
Affinity DataKi:  150nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169505(CHEMBL189809 | [9-(2-Bromo-4-isopropyl-phenyl)-2-t...)
Affinity DataKi:  150nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169539(Bis-cyclopropylmethyl-[9-(2,4-dichloro-phenyl)-2-t...)
Affinity DataKi:  240nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169534(CHEMBL187362 | Ethyl-phenethyl-[2-trifluoromethyl-...)
Affinity DataKi:  249nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169534(CHEMBL187362 | Ethyl-phenethyl-[2-trifluoromethyl-...)
Affinity DataKi:  249nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169522(CHEMBL188623 | Phenethyl-propyl-[2-trifluoromethyl...)
Affinity DataKi:  250nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169518((2,2,2-Trifluoro-ethyl)-[2-trifluoromethyl-9-(2,4,...)
Affinity DataKi:  291nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169512(CHEMBL360389 | Diphenethyl-[2-trifluoromethyl-9-(2...)
Affinity DataKi:  333nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169519(2-Methyl-9-(2,4,6-trimethyl-phenyl)-9H-benzo[d]imi...)
Affinity DataKi:  360nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169501((2-Cyclopropyl-ethyl)-propyl-[2-trifluoromethyl-9-...)
Affinity DataKi:  362nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169510(CHEMBL363218 | Cyclopropylmethyl-[9-(2,4-dichloro-...)
Affinity DataKi:  370nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169536(CHEMBL189798 | [9-(2-Bromo-4-isopropyl-phenyl)-2-t...)
Affinity DataKi:  410nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169506(Benzyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-pheny...)
Affinity DataKi:  428nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169504((2-Cyclopropyl-ethyl)-[2-trifluoromethyl-9-(2,4,6-...)
Affinity DataKi:  457nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169527(2-Ethyl-9-(2,4,6-trimethyl-phenyl)-9H-benzo[d]imid...)
Affinity DataKi:  570nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169499(Benzyl-methyl-[2-trifluoromethyl-9-(2,4,6-trimethy...)
Affinity DataKi:  573nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169516(CHEMBL365858 | Phenethyl-[2-trifluoromethyl-9-(2,4...)
Affinity DataKi:  618nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169502((2-Cyclopropyl-ethyl)-(2,2,2-trifluoro-ethyl)-[2-t...)
Affinity DataKi:  653nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169500(Butyl-ethyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-...)
Affinity DataKi:  704nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169525(CHEMBL364809 | Phenethyl-(2,2,2-trifluoro-ethyl)-[...)
Affinity DataKi:  744nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169514(2-Ethyl-6-fluoro-9-(2,4,6-trimethyl-phenyl)-9H-ben...)
Affinity DataKi:  930nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169530(6-Fluoro-2-methyl-9-(2,4,6-trimethyl-phenyl)-9H-be...)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169538((2-Cyclopropyl-ethyl)-ethyl-[2-trifluoromethyl-9-(...)
Affinity DataKi:  1.41E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169528(CHEMBL362124 | [9-(2,4-Dichloro-phenyl)-2-trifluor...)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169503(Benzyl-ethyl-[2-trifluoromethyl-9-(2,4,6-trimethyl...)
Affinity DataKi:  2.77E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169532(2-Trifluoromethyl-9-(2,4,6-trimethyl-phenyl)-9H-be...)
Affinity DataKi:  3.56E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169513(Benzyl-propyl-[2-trifluoromethyl-9-(2,4,6-trimethy...)
Affinity DataKi:  4.05E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169521(Benzyl-butyl-[2-trifluoromethyl-9-(2,4,6-trimethyl...)
Affinity DataKi:  7.71E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed