Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50016908
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universidade Do Porto

Curated by ChEMBL
LigandPNGBDBM50175102(1-(4-amino-2,3-dihydro-1,2,5-oxadiazol-3-yl)-5-(pi...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universidade Do Porto

Curated by ChEMBL
LigandPNGBDBM50175103(4-(5-(piperidin-1-ylmethyl)-4-(5-(pyridin-4-yl)-4H...)
Affinity DataIC50:  280nMAssay Description:Inhibitory activity against GSK3betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Universidade Do Porto

Curated by ChEMBL
LigandPNGBDBM50175102(1-(4-amino-2,3-dihydro-1,2,5-oxadiazol-3-yl)-5-(pi...)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibitory activity against CDK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Universidade Do Porto

Curated by ChEMBL
LigandPNGBDBM50175103(4-(5-(piperidin-1-ylmethyl)-4-(5-(pyridin-4-yl)-4H...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibitory activity against CDK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed