Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50000520
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006842(2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-3-(3-isopropox...)
Affinity DataIC50:  9.30nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006838(2-[2-(1H-Indol-3-yl)-ethyl]-3-(3-isopropoxy-phenyl...)
Affinity DataIC50:  26nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006839(2-[2-(1H-Indol-3-yl)-propyl]-3-(3-isopropoxy-pheny...)
Affinity DataIC50:  70nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006840(2-[2-(1H-Indol-3-yl)-vinyl]-3-(3-isopropoxy-phenyl...)
Affinity DataIC50:  430nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006837(2-[2-(1H-Indol-3-yl)-ethyl]-3-phenyl-3H-quinazolin...)
Affinity DataIC50:  670nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006836(2-[2-(5-Bromo-1H-indol-3-yl)-vinyl]-3-(3-isopropox...)
Affinity DataIC50:  1.40E+3nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006841(2-[2-(1H-Indol-3-yl)-1-methyl-ethyl]-3-(3-isopropo...)
Affinity DataIC50:  9.10E+3nMAssay Description:Evaluated for inhibition of [125I]-CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 microM (in vi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed