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Found 10 Enz. Inhib. hit(s) with all data for entry = 1466
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals

LigandPNGBDBM11558((3S)-2-[(3R)-3-amino-4-(2-fluorophenyl)butanoyl]-1...)
Affinity DataIC50:  23nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals

LigandPNGBDBM11559(N-({(2S)-1-[(3R)-3-amino-4-(2-fluorophenyl)butanoy...)
Affinity DataIC50:  90nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals

LigandPNGBDBM11464((2S,3S)-2-amino-3-methyl-1-(1,3-thiazolidin-3-yl)p...)
Affinity DataIC50:  140nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Santhera Pharmaceuticals

LigandPNGBDBM11559(N-({(2S)-1-[(3R)-3-amino-4-(2-fluorophenyl)butanoy...)
Affinity DataIC50:  410nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals

LigandPNGBDBM11557((2S)-1-[(3R)-3-amino-4-phenylbutanoyl]-N-({5-chlor...)
Affinity DataIC50:  1.90E+3nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | 1-METHYLAMINE-1...)
Affinity DataIC50:  3.00E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | 1-METHYLAMINE-1...)
Affinity DataIC50:  3.30E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Santhera Pharmaceuticals

LigandPNGBDBM11556(2-(2-chlorophenyl)-2-(morpholin-4-yl)ethan-1-amine...)
Affinity DataIC50:  3.30E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Santhera Pharmaceuticals

LigandPNGBDBM11556(2-(2-chlorophenyl)-2-(morpholin-4-yl)ethan-1-amine...)
Affinity DataIC50:  4.60E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Santhera Pharmaceuticals

LigandPNGBDBM11558((3S)-2-[(3R)-3-amino-4-(2-fluorophenyl)butanoyl]-1...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair