Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50017425
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181998(7-(pyridin-3-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182014(7-(pyridin-2-yl)-N-(3,4,5-trimethoxyphenyl)-6,7-di...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182013(5-bromo-N4-(pyridin-2-yl)-N2-(3,4,5-trimethoxyphen...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182006(8-(pyridin-2-yl)-2-(3,4,5-trimethoxyphenylamino)-5...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181975(8-(pyridin-2-yl)-N-(3,4,5-trimethoxyphenyl)-5,6,7,...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181987(CHEMBL204933 | ethyl 2-(4-(pyridin-2-ylamino)-2-(3...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182010(7-(pyridin-2-yl)-N-(2,4,6-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181983(CHEMBL377957 | N-(5-methoxy-2-methylphenyl)-7-(pyr...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181979(7-(4-methoxypyridin-3-yl)-N-(3,4,5-trimethoxypheny...)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181968(7-(pyridin-2-yl)-N-(5,6,7,8-tetrahydronaphthalen-1...)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182002(4-methyl-3-(7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyri...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181981(7-(4-chloropyridin-3-yl)-N-(3,4,5-trimethoxyphenyl...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181969(7-(pyridin-2-yl)-N-o-tolyl-7H-pyrrolo[2,3-d]pyrimi...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181999(7-(thiazol-2-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181982(CHEMBL208042 | N-(3-methoxyphenyl)-7-(pyridin-2-yl...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181986(CHEMBL206853 | N-(2-methyl-5-(quinoxalin-2-yl)phen...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182005(CHEMBL207935 | N-(2-chlorophenyl)-7-(pyridin-2-yl)...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182015(CHEMBL206322 | N-(2-methoxyphenyl)-7-(pyridin-2-yl...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182007(7-(pyridin-2-yl)-N-m-tolyl-7H-pyrrolo[2,3-d]pyrimi...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181988(7-(2-chloropyridin-4-yl)-N-(3,4,5-trimethoxyphenyl...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182018(7-(2-chloropyrimidin-4-yl)-N-(3,4,5-trimethoxyphen...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182012(7-(4-fluoropyridin-3-yl)-N-(3,4,5-trimethoxyphenyl...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181994(CHEMBL382637 | N-(2-ethylphenyl)-7-(pyridin-2-yl)-...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182009(CHEMBL381308 | N-(2-(methylthio)phenyl)-7-(pyridin...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182019(CHEMBL378596 | N-(2-fluorophenyl)-7-(pyridin-2-yl)...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181977(CHEMBL203020 | N-(2-bromophenyl)-7-(pyridin-2-yl)-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181966(CHEMBL381609 | N-(3-(methylthio)phenyl)-7-(pyridin...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181976(CHEMBL383834 | N-(5-iodo-2-methylphenyl)-7-(pyridi...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181973(7-(pyridin-2-yl)-N-(2-(trifluoromethyl)phenyl)-7H-...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182000(7-(2-(pyridin-4-yl)ethyl)-N-(3,4,5-trimethoxypheny...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181997(7-(pyridin-3-ylmethyl)-N-(3,4,5-trimethoxyphenyl)-...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181978(CHEMBL203676 | N-(4-iodo-2-methylphenyl)-7-(pyridi...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181990(7-(pyridin-4-yl)-N-(3,4,5-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182017(7-(pyridin-2-yl)-2-(3,4,5-trimethoxyphenylamino)-5...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182011(CHEMBL206796 | ethyl 2-(4-chloro-2-(3,4,5-trimetho...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182008(CHEMBL203675 | N-(5-bromo-2-methylphenyl)-7-(pyrid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182003(7-(2-(pyridin-3-yl)ethyl)-N-(3,4,5-trimethoxypheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182004(7-(pyridin-2-yl)-N-(4-(trifluoromethyl)phenyl)-7H-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182001(3-(7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181995(CHEMBL381998 | N-(3,4,5-trimethoxybenzyl)-7-(pyrid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181996(8-(pyridin-2-yl)-2-(3,4,5-trimethoxyphenylamino)py...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181993(1-(3-(7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181992(7-(4-chloropyrimidin-2-yl)-N-(3,4,5-trimethoxyphen...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181991((4-methyl-3-(7-(pyridin-2-yl)-7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181989(CHEMBL204982 | N-benzyl-7-(pyridin-2-yl)-7H-pyrrol...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181985(7-(5-methylpyridin-2-yl)-N-(3,4,5-trimethoxyphenyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181984(CHEMBL380116 | N-(2-isopropylphenyl)-7-(pyridin-2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181980(2-(4-methylpiperazin-1-yl)-7-(pyridin-2-yl)-7H-pyr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181974(CHEMBL208169 | N-(1H-indol-6-yl)-7-(pyridin-2-yl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50181972(CHEMBL205943 | N-(2-methyl-5-nitrophenyl)-7-(pyrid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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