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Found 10 Enz. Inhib. hit(s) with all data for entry = 50018316
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194321((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194319((E)-N-(4-chlorophenyl)-2-(3-ethyl-2-methyl-6,7-dih...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194318((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194325((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...)
Affinity DataIC50:  280nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194324((E)-N-(4-acetylphenyl)-2-(2,3-diethyl-1-methyl-6,7...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194317((E)-N-(4-chlorophenyl)-2-(2,3-dimethyl-6,7-dihydro...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194322((E)-N-(4-chlorophenyl)-2-(3-ethyl-2-methyl-6,7-dih...)
Affinity DataIC50:  440nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194323((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...)
Affinity DataIC50:  750nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194320((E)-N-(4-chlorophenyl)-2-(6,7-dihydro-1H-indol-4(5...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Kv1.5 expressed in LTK- cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194321((E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of hERG expressed in HEK cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed