Compile Data Set for Download or QSAR
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Found 96 Enz. Inhib. hit(s) with all data for entry = 50018850
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056569(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50118599(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  0.710nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50118600(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperid...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50183539(CHEMBL381256 | CHEMBL429492 | trans-(R,R)-4-[2-[bi...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM22199(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-[(2E)-3-...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50118606(1-(benzofuran-2-ylmethyl)-4-(2-(bis(4-fluorophenyl...)
Affinity DataKi:  1.01nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126823(1-(4-bromobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126814(1-(4-(trifluoromethyl)benzyl)-4-(2-(bis(4-fluoroph...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126817(4-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperid...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126820(1-(4-nitrobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126813(1-(4-chlorobenzyl)-4-(2-(bis(4-fluorophenyl)methox...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50183547(CHEMBL206128 | CHEMBL255065 | trans-(S,S)-4-[2-[bi...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126386((1R,2S)-2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50118604(1-(benzo[b]thiophen-2-ylmethyl)-4-(2-(bis(4-fluoro...)
Affinity DataKi:  1.61nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126815(1-(4-iodobenzyl)-4-(2-(bis(4-fluorophenyl)methoxy)...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126822(1-(4-fluorobenzyl)-4-(2-(bis(4-fluorophenyl)methox...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126349(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  2.96nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126352((1R,2S)-2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056568(1-(benzo[b]thiophen-2-ylmethyl)-4-(2-(bis(4-fluoro...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199746((S)-3-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pip...)
Affinity DataKi:  4.77nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50118603(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(3-pheny...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126816(4-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-1-(4-m...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM22200(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3,4-dih...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056551(1-(benzofuran-2-ylmethyl)-4-(2-(bis(4-fluorophenyl...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126819(1-(4-methoxybenzyl)-4-(2-(bis(4-fluorophenyl)metho...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056571(1-(2-(bis(4-fluorophenyl)methoxy)ethyl)-4-(naphtha...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199741((R)-3-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pip...)
Affinity DataKi:  9.32nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50049365(1-Benzyl-4-{2-[bis-(4-fluoro-phenyl)-methoxy]-ethy...)
Affinity DataKi:  9.90nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126818(1-(3-methoxybenzyl)-4-(2-(bis(4-fluorophenyl)metho...)
Affinity DataKi:  13.3nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126352((1R,2S)-2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199741((R)-3-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pip...)
Affinity DataKi:  15.2nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50118602(4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(naphtha...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056577(3-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  16.1nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199737((1R,2R)-2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199742(1-(2-(bis(4-fluorophenyl)methoxy)ethyl)-4-(3-pheny...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50183539(CHEMBL381256 | CHEMBL429492 | trans-(R,R)-4-[2-[bi...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126349(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126386((1R,2S)-2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056581(1-(2-(bis(4-fluorophenyl)methoxy)ethyl)-4-(naphtha...)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199737((1R,2R)-2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50123386(1-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-4-ethy...)
Affinity DataKi:  33.7nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50123385(1-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-4-prop...)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199747(1-(2-(bis(4-fluorophenyl)methoxy)ethyl)-4-(3-chlor...)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50199746((S)-3-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)pip...)
Affinity DataKi:  48.1nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126348(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056578(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  51nMAssay Description:Displacement of [125I]RTI55 from SERT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126359(1-(2-(bis(4-fluorophenyl)methoxy)ethyl)-4-((6-meth...)
Affinity DataKi:  53nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50056578(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  56nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Heights

Curated by ChEMBL
LigandPNGBDBM50126370(2-((4-(2-(bis(4-fluorophenyl)methoxy)ethyl)piperaz...)
Affinity DataKi:  57nMAssay Description:Displacement of [125I]RTI55 from DAT in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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