Compile Data Set for Download or QSAR
maximum 50k data
Found 160 Enz. Inhib. hit(s) with all data for entry = 50041839
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM5815(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8826(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}phenyl)-1...)
Affinity DataIC50:  3.02nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8870(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}phenyl)-1...)
Affinity DataIC50:  3.02nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM5815(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50:  3.02nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8813(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  6.03nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8826(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}phenyl)-1...)
Affinity DataIC50:  6.03nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8813(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  8.91nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8862(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-3-fluoro...)
Affinity DataIC50:  11.0nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8844(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  12.0nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8867(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-2-methox...)
Affinity DataIC50:  12.9nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8833(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  15.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8860(3-{4-[4-amino-6-(3-hydroxypropyl)thieno[2,3-d]pyri...)
Affinity DataIC50:  15.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8847(3-[4-amino-5-(4-{[(3-methylphenyl)carbamoyl]amino}...)
Affinity DataIC50:  17.0nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8846(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  17.0nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8844(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  19.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8858(3-{4-[4-amino-6-(2-hydroxyethyl)thieno[2,3-d]pyrim...)
Affinity DataIC50:  19.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8832(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  19.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8865(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-2-fluoro...)
Affinity DataIC50:  19.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8838(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  21.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM5816(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50:  21.9nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8860(3-{4-[4-amino-6-(3-hydroxypropyl)thieno[2,3-d]pyri...)
Affinity DataIC50:  25.7nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8824(3-(4-{4-amino-6-ethylthieno[2,3-d]pyrimidin-5-yl}p...)
Affinity DataIC50:  26.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8853(3-(4-{4-amino-6-propylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  26.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8835(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  26.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8862(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-3-fluoro...)
Affinity DataIC50:  26.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8867(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-2-methox...)
Affinity DataIC50:  28.2nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8824(3-(4-{4-amino-6-ethylthieno[2,3-d]pyrimidin-5-yl}p...)
Affinity DataIC50:  28.2nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM5814(3-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50:  28.2nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8839(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  28.8nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8812(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  32.4nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8836(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  33.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8856(3-{4-[4-amino-6-(pyridin-3-ylmethyl)thieno[2,3-d]p...)
Affinity DataIC50:  33.9nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM50416743(CHEMBL372744)
Affinity DataIC50:  33.9nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8838(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  34.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8832(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  34.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM5810(N-{3-[4-amino-5-(4-phenylphenyl)furo[2,3-d]pyrimid...)
Affinity DataIC50:  36.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8812(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  36.3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8858(3-{4-[4-amino-6-(2-hydroxyethyl)thieno[2,3-d]pyrim...)
Affinity DataIC50:  37.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8865(3-(4-{4-aminothieno[2,3-d]pyrimidin-5-yl}-2-fluoro...)
Affinity DataIC50:  38.0nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8843(Methyl 3-[({[4-(4-Amino-6-methylthieno[2,3-d]pyrim...)
Affinity DataIC50:  42.7nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8840(-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-...)
Affinity DataIC50:  45.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8846(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  45.7nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8841(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  47.9nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8831(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  50.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8869(3-(4-{4-amino-6-ethylthieno[2,3-d]pyrimidin-5-yl}p...)
Affinity DataIC50:  50.1nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8840(-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-...)
Affinity DataIC50:  50.1nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8830(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8857(3-{4-[4-amino-6-(pyridin-4-ylmethyl)thieno[2,3-d]p...)
Affinity DataIC50:  52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8836(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8842(3-(4-{4-amino-6-methylthieno[2,3-d]pyrimidin-5-yl}...)
Affinity DataIC50:  52.5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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