TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 30 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 3000 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 7.10E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 8.90E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 9.80E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-2(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Activity at human alpha2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair