Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50037915
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214016(CHEMBL243342 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214007(CHEMBL394621 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214001(CHEMBL389494 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  290nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214008(CHEMBL243343 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214003(CHEMBL243134 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  390nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214000(CHEMBL243180 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  450nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214004(CHEMBL243116 | N-(4-((1-(2-fluorobenzyl)-3-butyl-2...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214014(CHEMBL245018 | N-(4-((1-(2-fluorobenzyl)-3-butyl-2...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214010(CHEMBL244165 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  690nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214012(CHEMBL394368 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  790nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214009(3-(cyclopropylmethyl)-8-({4-[(dimethylsulfamoyl)am...)
Affinity DataIC50:  960nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214002(CHEMBL244590 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214015(1-(2-fluorobenzyl)-8-(4-aminobenzyl)-3-(cyclopropy...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214006(CHEMBL397513 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214013(CHEMBL242486 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214017(CHEMBL244589 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataIC50:  2.07E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50133801(CHEMBL120708 | N-(4-((1-(2-fluorobenzyl)-3-butyl-2...)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214018(CHEMBL428567 | N-(4-((1-(2-fluorobenzyl)-3-butyl-2...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214011(1-(2-fluorobenzyl)-8-(4-aminobenzyl)-3-butyl-1H-pu...)
Affinity DataIC50:  2.56E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214019(8-(2,4-diaminobenzyl)-1-(2-fluorobenzyl)-3-butyl-1...)
Affinity DataIC50:  5.65E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214005(CHEMBL242437 | N-{3-acetylamino-4-[3-butyl-1-(2-fl...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of human cPEPCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214016(CHEMBL243342 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataEC50:  8.20E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214010(CHEMBL244165 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataEC50:  4.70E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214012(CHEMBL394368 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214004(CHEMBL243116 | N-(4-((1-(2-fluorobenzyl)-3-butyl-2...)
Affinity DataEC50:  3.97E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50133801(CHEMBL120708 | N-(4-((1-(2-fluorobenzyl)-3-butyl-2...)
Affinity DataEC50:  8.60E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214001(CHEMBL389494 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataEC50:  2.17E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214007(CHEMBL394621 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataEC50:  5.57E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214013(CHEMBL242486 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataEC50:  5.50E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50214003(CHEMBL243134 | N-(4-((1-(2-fluorobenzyl)-3-(cyclop...)
Affinity DataEC50:  8.75E+3nMAssay Description:Inhibition of cPEPCK in rat H4IIE cells assessed as effect on glucose productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed