Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 3048
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27251(indan derivative, 1 | tert-butyl 2-(2-benzenesulfo...)
Affinity DataEC50:  190nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  15nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27253(Boc-indole derivative, 11 | tert-butyl 2-[4-(2-ben...)
Affinity DataEC50:  120nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27254(Boc-indole derivative, 12 | tert-butyl 2-[4-(benze...)
Affinity DataEC50:  220nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27255(Boc-indole derivative, 13 | tert-butyl 2-[4-(3-ben...)
Affinity DataEC50:  350nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27256(Boc-indole derivative, 14 | tert-butyl 2-(4-benzen...)
Affinity DataEC50:  1.32E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27257(Boc-indole derivative, 15 | tert-butyl 2-{4-[2-(th...)
Affinity DataEC50:  58nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27258(Boc-indole derivative, 16 | tert-butyl 2-[4-(2-{[5...)
Affinity DataEC50:  230nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27259(Boc-indole derivative, 17 | tert-butyl 2-{4-[(phen...)
Affinity DataEC50:  1.80E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27260(Boc-indole derivative, 18 | tert-butyl 2-{4-[2-(ph...)
Affinity DataEC50:  1.75E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27261(Boc-indole derivative, 19 | tert-butyl 2-{4-[3-(ph...)
Affinity DataEC50:  360nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27262(Boc-indole derivative, 20 | tert-butyl 2-[4-(amino...)
Affinity DataEC50:  5.60E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27263(Boc-indole derivative, 21 | tert-butyl 2-[4-(cyano...)
Affinity DataEC50:  300nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27264(Boc-indole derivative, 22 | tert-butyl 2-[4-(2-cya...)
Affinity DataEC50:  130nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27265(Boc-indole derivative, 23 | tert-butyl 2-[4-(3-hyd...)
Affinity DataEC50:  380nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27266(Boc-indole derivative, 24 | tert-butyl 2-[4-(2-hyd...)
Affinity DataEC50:  420nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27267(3-(4-{1-[(tert-butoxy)carbonyl]-1H-indol-2-yl}phen...)
Affinity DataEC50:  220nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27268(Boc-indole derivative, 26 | tert-butyl 2-[4-(2-car...)
Affinity DataEC50:  57nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27269(Boc-indole derivative, 27 | tert-butyl 2-{4-[(1E)-...)
Affinity DataEC50:  4.90E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27270(Boc-indole derivative, 28 | tert-butyl 2-{4-[2-(me...)
Affinity DataEC50:  490nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27271(Boc-indole derivative, 29 | tert-butyl 2-(4-{2-[(2...)
Affinity DataEC50:  1.51E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27272(Boc-indole derivative, 30 | tert-butyl 2-{4-[2-(ph...)
Affinity DataEC50:  1.78E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27273(3-[4-(1-benzoyl-1H-indol-2-yl)phenyl]propanenitril...)
Affinity DataEC50:  12nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27274(N-{2-[4-(1-benzoyl-1H-indol-2-yl)phenyl]ethyl}benz...)
Affinity DataEC50:  1.78E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27251(indan derivative, 1 | tert-butyl 2-(2-benzenesulfo...)
Affinity DataEC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27264(Boc-indole derivative, 22 | tert-butyl 2-[4-(2-cya...)
Affinity DataEC50:  1.19E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27267(3-(4-{1-[(tert-butoxy)carbonyl]-1H-indol-2-yl}phen...)
Affinity DataEC50:  1.15E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27268(Boc-indole derivative, 26 | tert-butyl 2-[4-(2-car...)
Affinity DataEC50:  1.11E+3nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27273(3-[4-(1-benzoyl-1H-indol-2-yl)phenyl]propanenitril...)
Affinity DataEC50:  220nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM19992(2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methy...)
Affinity DataEC50:  367nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  40nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM19992(2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methy...)
Affinity DataEC50:  35nMAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Tanabe Research Laboratories Usa

LigandPNGBDBM27252(Boc-indole derivative, 10 | tert-butyl 2-[3-(2-ben...)
Affinity DataEC50:  420nMpH: 7.5 T: 2°CAssay Description:Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed