Compile Data Set for Download or QSAR
maximum 50k data
Found 79 Enz. Inhib. hit(s) with all data for entry = 50020824
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218023(CHEMBL248734 | {[2-(5-benzo[1,3]dioxol-5-yl-2'-chl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218032(({2-[2'-chloro-5-(2,3-dihydro-benzofuran-5-yl)-bip...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218017(({2-[2'-chloro-5-(2,3-dihydro-benzo[1,4]dioxin-6-y...)
Affinity DataIC50:  14nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218012(({2-[4-(2,3-dihydro-benzofuran-5-yl)-2-thiophen-2-...)
Affinity DataIC50:  17nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218004(({2-[4'-methoxy-3'-methyl-3-(thiophene-2-carbonyl)...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218001(({2-[4-benzo[1,3]dioxol-5-yl-2-(thiophene-2-carbon...)
Affinity DataIC50:  19nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218016(({2-[4-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-2-thiop...)
Affinity DataIC50:  25nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218007(({2-[3'-chloro-3-(thiophene-2-carbonyl)-biphenyl-4...)
Affinity DataIC50:  26nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218021(({2-[4'-methoxy-3-(thiophene-2-carbonyl)-biphenyl-...)
Affinity DataIC50:  27nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218005(CHEMBL251775 | {[2-(2''-chloro-4-methoxy-3-methyl-...)
Affinity DataIC50:  28nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218002(CHEMBL401191 | {[2-(4-benzo[1,3]dioxol-5-yl-2-thio...)
Affinity DataIC50:  34nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218014(CHEMBL250372 | {methyl-[2-(3-thiophen-2-ylmethyl-b...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217995((methyl-{2-[3-(thiophene-2-carbonyl)-biphenyl-4-yl...)
Affinity DataIC50:  45nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218003((methyl-{2-[3'-methyl-3-(thiophene-2-carbonyl)-bip...)
Affinity DataIC50:  45nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218022(CHEMBL404856 | {[2-(2''-chloro-[1,1';3',1'']terphe...)
Affinity DataIC50:  53nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217996(CHEMBL248920 | {methyl-[2-(2''-methyl-[1,1';3',1''...)
Affinity DataIC50:  56nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218033((methyl-{2-[4'-methyl-3-(thiophene-2-carbonyl)-bip...)
Affinity DataIC50:  59nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217998(CHEMBL401422 | {[2-(3-benzoyl-biphenyl-4-yloxy)-et...)
Affinity DataIC50:  65nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217997(({2-[4'-chloro-3-(thiophene-2-carbonyl)-biphenyl-4...)
Affinity DataIC50:  68nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218030(CHEMBL250373 | {methyl-[2-(3-thiophen-2-yl-bipheny...)
Affinity DataIC50:  70nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218009(CHEMBL250581 | {[2-(3-cyclohexanecarbonyl-biphenyl...)
Affinity DataIC50:  70nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218025(({2-[3',4'-dimethyl-3-(thiophene-2-carbonyl)-biphe...)
Affinity DataIC50:  76nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218028(CHEMBL250374 | {[2-(3-benzyl-biphenyl-4-yloxy)-eth...)
Affinity DataIC50:  85nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218029(({2-[3'-methoxy-3-(thiophene-2-carbonyl)-biphenyl-...)
Affinity DataIC50:  104nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218000(CHEMBL251150 | {[2-(2''-fluoro-[1,1';3',1'']terphe...)
Affinity DataIC50:  108nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218026(CHEMBL249126 | {methyl-[2-(3-thiophen-3-yl-bipheny...)
Affinity DataIC50:  139nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218013(CHEMBL400979 | {[2-(4'-methoxy-3'-methyl-3-thiophe...)
Affinity DataIC50:  161nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218027(({2-[2'-chloro-3-(thiophene-2-carbonyl)-biphenyl-4...)
Affinity DataIC50:  175nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218020(CHEMBL250580 | {methyl-[2-([1,1';3',1'']terphenyl-...)
Affinity DataIC50:  229nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217999(CHEMBL250582 | {[2-(3-cyclohexyl-biphenyl-4-yloxy)...)
Affinity DataIC50:  251nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218024(CHEMBL399983 | {[2-(3-cyclohexylmethyl-biphenyl-4-...)
Affinity DataIC50:  289nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218018(CHEMBL249125 | {[2-(2''-methoxy-[1,1';3',1'']terph...)
Affinity DataIC50:  351nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218011(CHEMBL250356 | {methyl-[2-(3-naphthalen-1-yl-biphe...)
Affinity DataIC50:  496nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218006((methyl-{2-[2'-methyl-3-(thiophene-2-carbonyl)-bip...)
Affinity DataIC50:  632nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218031(CHEMBL250784 | {[2-(3''-chloro-[1,1';3',1'']terphe...)
Affinity DataIC50:  674nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218015((methyl-{2-[2-(thiophene-2-carbonyl)-4-trifluorome...)
Affinity DataIC50:  702nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218019(({2-[3',4'-dimethoxy-3-(thiophene-2-carbonyl)-biph...)
Affinity DataIC50:  834nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218010(CHEMBL250152 | {methyl-[2-(3-thiazol-2-yl-biphenyl...)
Affinity DataIC50:  957nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218008(CHEMBL399144 | {[2-(4''-chloro-[1,1';3',1'']terphe...)
Affinity DataIC50:  965nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT1 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218024(CHEMBL399983 | {[2-(3-cyclohexylmethyl-biphenyl-4-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218009(CHEMBL250581 | {[2-(3-cyclohexanecarbonyl-biphenyl...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217999(CHEMBL250582 | {[2-(3-cyclohexyl-biphenyl-4-yloxy)...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218008(CHEMBL399144 | {[2-(4''-chloro-[1,1';3',1'']terphe...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218000(CHEMBL251150 | {[2-(2''-fluoro-[1,1';3',1'']terphe...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218032(({2-[2'-chloro-5-(2,3-dihydro-benzofuran-5-yl)-bip...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218012(({2-[4-(2,3-dihydro-benzofuran-5-yl)-2-thiophen-2-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218027(({2-[2'-chloro-3-(thiophene-2-carbonyl)-biphenyl-4...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50218018(CHEMBL249125 | {[2-(2''-methoxy-[1,1';3',1'']terph...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217995((methyl-{2-[3-(thiophene-2-carbonyl)-biphenyl-4-yl...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50217996(CHEMBL248920 | {methyl-[2-(2''-methyl-[1,1';3',1''...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of [14C]glycine reuptake at human GlyT2 expressed in BE(2)-C cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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