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Found 21 Enz. Inhib. hit(s) with all data for entry = 50038460
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(CHEMBL443683 | telomestatin)
Affinity DataIC50:  0.640nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(CHEMBL443683 | telomestatin)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50134030(9-[4-(N,N-dimethylamino)phenylamino]-3,6-bis(3-pyr...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50:  45nMAssay Description:Inhibition of human telomerase expressed in in HEK293T cells in presence of primer (T2AG3)4 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50:  52nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(CHEMBL443683 | telomestatin)
Affinity DataIC50:  58nMAssay Description:Inhibition of human telomerase expressed in in HEK293T cells in presence of primer (T2AG3)4 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50:  63nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  63nMAssay Description:Inhibition of human telomerase expressed in in HEK293T cells in presence of primer (T2AG3)4 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50134030(9-[4-(N,N-dimethylamino)phenylamino]-3,6-bis(3-pyr...)
Affinity DataIC50:  65nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated before telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  710nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50107609(5,10,15,20-tetra(1-methyl-4-pyridyl)-porphyrin | C...)
Affinity DataIC50:  740nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells treated after telomerase elongation by telomeric repeat amplification protocol assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  790nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50134030(9-[4-(N,N-dimethylamino)phenylamino]-3,6-bis(3-pyr...)
Affinity DataIC50:  830nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(CHEMBL443683 | telomestatin)
Affinity DataIC50:  900nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50339190(CHEMBL443683 | telomestatin)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer TS by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376748(CHEMBL259739 | Phen-DC3)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer TS by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer (T2AG3)3 by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Institut National De La Sant£

Curated by ChEMBL
LigandPNGBDBM50376747(CHEMBL409247)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of human telomerase expressed in HEK293T cells in presence of primer TS by primer extension assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed