Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 4615
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Munich

LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Munich

LigandPNGBDBM50218894(7-bromoindirubin-3-oxime | 7BIO | CHEMBL1092509)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Munich

LigandPNGBDBM7393(3-[(2Z,3E)-3-(hydroxyimino)-2,3-dihydro-1H-indol-2...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Munich

LigandPNGBDBM81296(5BIO)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed