Found 89 Enz. Inhib. hit(s) with all data for entry = 50042281 
Affinity DataKd: 182nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 5.62E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 1.78E+4nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 7.24E+3nMAssay Description:Binding affinity to human recombinant sst3 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.63E+3nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 1.20nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 6.46E+3nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.32E+4nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 8.13E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 4.90E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 56nMAssay Description:Binding affinity to human dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.603nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 1.48E+3nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 0.759nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 0.380nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+4nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 2.95E+3nMAssay Description:Binding affinity to human recombinant sst3 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.30nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 1.23E+4nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.95E+4nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 50nMAssay Description:Binding affinity to human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKd: 7.94E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 7.76E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 0.372nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 3.89E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 3.02E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 9.33E+3nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.204nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 8.13E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 5.62E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.372nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 0.977nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 6.46E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 123nMAssay Description:Binding affinity to human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 1.95E+3nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 501nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 7.24E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 5.62E+4nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKd: 28nMAssay Description:Binding affinity to human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKd: 8.51E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 0.282nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKd: 4.90E+4nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
