Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50026178
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270672(CHEMBL509847 | N1-(1-(4-(1H-Indazol-3-yl)phenyl)-1...)
Affinity DataIC50:  20nMAssay Description:Displacement of biotin-labeled pep-JIP1 from GST fused JNK1 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270672(CHEMBL509847 | N1-(1-(4-(1H-Indazol-3-yl)phenyl)-1...)
Affinity DataIC50:  295nMAssay Description:Inhibition of JNK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270641(CHEMBL528100 | N-(4-(1-Oxo-2,2,6,6-tetramethylpipe...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of JNK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270670(4-(4-(1H-Indazol-3-yl)benzamido)butanoic acid | CH...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of JNK1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270671(Ac-RPTTLNL-OH | CHEMBL504550)
Affinity DataIC50:  5.30E+4nMAssay Description:Displacement of biotin-labeled pep-JIP1 from GST fused JNK1 (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed