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Found 12 Enz. Inhib. hit(s) with all data for entry = 5622
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91713(Androst-4-en-3,17-dione, 2 | Androst-4-ene-3,17-di...)
Affinity DataIC50:  1.55E+3nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  8.50E+3nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91719(1-Dehydrotestosterone, 8)
Affinity DataIC50:  2.09E+4nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM8885((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...)
Affinity DataIC50:  5.35E+4nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91722(11alpha-17beta-Dihydroxyandrost-1,4-dien-3-one, 11)
Affinity DataIC50:  6.15E+4nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91721(11alpha-Hydroxytestosterone, 10)
Affinity DataIC50:  8.90E+4nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91715(17beta-Hydroxy-5alpha-androstan-3,6-dione, 4)
Affinity DataIC50:  9.59E+4nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91718(Androst-1,4-dien-3,17-dione, 7)
Affinity DataIC50:  1.03E+5nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91716(11alpha-Hydroxyandrost-4-en-3,17-dione, 5)
Affinity DataIC50:  1.41E+5nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91714(Testolactone, 3)
Affinity DataIC50:  1.42E+5nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91720(11alpha-Hydroxyandrost-1,4-dien-3,17-dione, 9)
Affinity DataIC50:  1.65E+5nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Jordan

LigandPNGBDBM91717(11alpha-Hydroxytestolactone, 6)
Affinity DataIC50:  2.84E+5nMAssay Description:AChE and BChE inhibiting activities were measured in vitro by a modified spectrophotometric method previously developed by Ellman et. al.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed