Compile Data Set for Download or QSAR
maximum 50k data
Found 102 Enz. Inhib. hit(s) with all data for entry = 50027455
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246088(2-methyl-2-[2-methyl-4-({[1-methyl-5-(2'-methyl-bi...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at mouse PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  2.83E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  9.71E+3nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28710(2-[4-({[2-(4-tert-butylphenyl)-4-methyl-1,3-thiazo...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28710(2-[4-({[2-(4-tert-butylphenyl)-4-methyl-1,3-thiazo...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM28710(2-[4-({[2-(4-tert-butylphenyl)-4-methyl-1,3-thiazo...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246475(2-(4-((3-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246475(2-(4-((3-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246523(2-(4-((5-(4-tert-butylphenyl)-1H-pyrazole-3-carbox...)
Affinity DataEC50:  383nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246523(2-(4-((5-(4-tert-butylphenyl)-1H-pyrazole-3-carbox...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246523(2-(4-((5-(4-tert-butylphenyl)-1H-pyrazole-3-carbox...)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246524(2-(4-((3-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246524(2-(4-((3-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  2.17E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246524(2-(4-((3-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246525(2-(4-((5-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246525(2-(4-((5-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246525(2-(4-((5-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246526(2-(4-((3-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246526(2-(4-((3-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50246526(2-(4-((3-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245782(2-(4-((5-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245782(2-(4-((5-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  4.85E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245782(2-(4-((5-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245783(2-(4-((3-(4-isobutylphenyl)-1-methyl-1H-pyrazole-5...)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245783(2-(4-((3-(4-isobutylphenyl)-1-methyl-1H-pyrazole-5...)
Affinity DataEC50:  2.87E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245783(2-(4-((3-(4-isobutylphenyl)-1-methyl-1H-pyrazole-5...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245784(2-(4-((5-(4-isobutylphenyl)-1-methyl-1H-pyrazole-3...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245784(2-(4-((5-(4-isobutylphenyl)-1-methyl-1H-pyrazole-3...)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245784(2-(4-((5-(4-isobutylphenyl)-1-methyl-1H-pyrazole-3...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245785(2-(4-((3-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245785(2-(4-((3-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245785(2-(4-((3-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245843(2-(4-((5-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245843(2-(4-((5-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245843(2-(4-((5-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245944(2-(4-((1-allyl-3-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245944(2-(4-((1-allyl-3-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245944(2-(4-((1-allyl-3-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245945(2-(4-((1-allyl-5-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245945(2-(4-((1-allyl-5-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245945(2-(4-((1-allyl-5-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245946(2-(4-((3-(4-tert-butylphenyl)-1-(2-methoxyethyl)-1...)
Affinity DataEC50:  66nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245946(2-(4-((3-(4-tert-butylphenyl)-1-(2-methoxyethyl)-1...)
Affinity DataEC50:  2.05E+3nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245946(2-(4-((3-(4-tert-butylphenyl)-1-(2-methoxyethyl)-1...)
Affinity DataEC50:  303nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245947(2-(4-((5-(4-tert-butylphenyl)-1-(2-methoxyethyl)-1...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245947(2-(4-((5-(4-tert-butylphenyl)-1-(2-methoxyethyl)-1...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245947(2-(4-((5-(4-tert-butylphenyl)-1-(2-methoxyethyl)-1...)
Affinity DataEC50:  478nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245990(2-(4-((5-(4-tert-butylphenyl)-1-(2-morpholinoethyl...)
Affinity DataEC50:  570nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50245990(2-(4-((5-(4-tert-butylphenyl)-1-(2-morpholinoethyl...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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