Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50027508
TargetPeptidylglycine alpha-amidating monooxygenase(Rattus norvegicus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50273316(CHEMBL509495 | N-dansyl-Tyr-Val-D-Ala)
Affinity DataKi:  4.70E+5nMAssay Description:Inhibition of rat recombinant peptidylglycine alpha-amidating monooxygenase assessed as inhibition of N-dansyl-Tyr-Val-Gly amidationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidylglycine alpha-amidating monooxygenase(Rattus norvegicus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50273962(CHEMBL445286 | Phenylthioacetylglycine)
Affinity DataKi:  3.80E+6nMAssay Description:Inhibition of rat recombinant peptidylglycine alpha-amidating monooxygenase assessed as inhibition of N-dansyl-Tyr-Val-Gly amidationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidylglycine alpha-amidating monooxygenase(Rattus norvegicus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50273494(6-O-Palmitoyl-L-ascorbate | CHEMBL457018)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of rat recombinant peptidylglycine alpha-amidating monooxygenase in presence of DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed