Affinity DataKi: 2.51nMAssay Description:Displacement of [3H]PGE2 from EP1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 31.6nMAssay Description:Antagonist activity at EP1 receptor assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Binding affinity to TP receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Activity at EP3 receptor by FLIPR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.31nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12.6nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Rattus norvegicus (Rat))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 12.6nMAssay Description:Binding affinity to rat EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15.8nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Binding affinity to human EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Displacement of [3H]PGE2 from EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity to EP1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Activity at TP receptor by FLIPR methodMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Activity at PGF2alpha receptor by FLIPR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: >3.16E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG receptor by FLIPR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair