Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50027899
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277112(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50:  1nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277111(3-Benzo[1,3]dioxol-5-yl-3-[1-oxo-6-(1,2,3,4-tetrah...)
Affinity DataIC50:  2nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277112(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50:  5nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277098(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50:  7nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277111(3-Benzo[1,3]dioxol-5-yl-3-[1-oxo-6-(1,2,3,4-tetrah...)
Affinity DataIC50:  14nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277096(3-(6-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  39nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277111(3-Benzo[1,3]dioxol-5-yl-3-[1-oxo-6-(1,2,3,4-tetrah...)
Affinity DataIC50:  167nMAssay Description:Binding affinity to human integrin alpha2beta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277095(3-(5-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  180nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277075(3-(4-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  230nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277098(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50:  310nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277112(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50:  323nMAssay Description:Binding affinity to human integrin alpha2beta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277097(3-(7-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  370nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277096(3-(6-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  600nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277075(3-(4-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  2.05E+3nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277097(3-(7-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  4.30E+3nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277095(3-(5-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50:  4.80E+3nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277098(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50:  6.30E+3nMAssay Description:Binding affinity to human integrin alpha2beta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277097(3-(7-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human integrin alpha2beta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277095(3-(5-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human integrin alpha2beta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50277096(3-(6-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human integrin alpha2beta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed