Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50028744
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258290(1-[5,6-Dideoxy-6-[(hydroxypyrophosphoroxy)phosphon...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258291(9-[5'-Deoxy-5'-[(hydroxyphosphoroxy)phosphinyl]-be...)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258427(CHEMBL522015 | uridine5'-methylene-phosphonate)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258291(9-[5'-Deoxy-5'-[(hydroxyphosphoroxy)phosphinyl]-be...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM2(({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-...)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258288(9-[5'-Deoxy-5'-[(hydroxypyrophosphoroxy)phosphinyl...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50258289(9-[5'-Deoxy-5'-[(hydroxypyrophosphoroxy)phosphinyl...)
Affinity DataEC50:  8.60E+3nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells coexpressing phospholipase C-activating G protein assessed as inositol phosph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed